sample_idx
int64
503k
560k
fold
stringclasses
1 value
smiles
stringlengths
11
317
adduct
stringclasses
11 values
precursor_type
null
ionmode
null
precursor_mz
float64
115
1.47k
collision_energy
float64
15
75
instrument_type
null
spectrum_id
null
rank
int64
1
31.5k
n_candidates
int64
2
31.5k
gt_score
float64
-0.36
0.72
top1_smiles
stringlengths
8
317
top1_score
float64
-0.31
0.74
top_candidates
listlengths
2
50
top_scores
listlengths
2
50
method
stringclasses
4 values
display_name
stringclasses
4 values
score_semantics
stringclasses
1 value
zero_spectrum_embedding
int64
0
0
⌀
tie_break_rule
stringclasses
1 value
n_top_score_ties
int64
1
3
⌀
502,647
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
20
null
null
21
548
0.100249
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.136963
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CC(COC1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CCOC(C1)C2=C(OC(...
[ 0.1369626373052597, 0.13405099511146545, 0.1319037824869156, 0.13094200193881989, 0.12968526780605316, 0.12799321115016937, 0.1252405196428299, 0.12451738864183426, 0.12437218427658081, 0.1218419075012207, 0.11946996301412582, 0.11830828338861465, 0.11668667197227478, 0.11393295228481293, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,648
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
20
null
null
22
548
0.096242
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.13721
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1CC(CO1)C2=NC(=C...
[ 0.13721048831939697, 0.13413546979427338, 0.13224709033966064, 0.13138899207115173, 0.12850181758403778, 0.12710173428058624, 0.1250784695148468, 0.12502579391002655, 0.12296164035797119, 0.12137569487094879, 0.11914234608411789, 0.11174221336841583, 0.11156905442476273, 0.1108043268322944...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,649
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
60
null
null
24
548
0.100622
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.132645
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1CC(CO1)C2=NC(=C...
[ 0.13264499604701996, 0.13002946972846985, 0.12636874616146088, 0.12616737186908722, 0.12410686910152435, 0.12079635262489319, 0.12074214220046997, 0.12044796347618103, 0.11910523474216461, 0.11860018968582153, 0.11698532104492188, 0.11617645621299744, 0.11494007706642151, 0.107951782643795...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,650
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
30
null
null
23
548
0.09448
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.127686
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.12768560647964478, 0.12705948948860168, 0.1246514543890953, 0.12404081970453262, 0.12172451615333557, 0.11674667149782181, 0.11124938726425171, 0.10850436985492706, 0.10783903300762177, 0.10487999022006989, 0.10455136001110077, 0.10342217981815338, 0.10293052345514297, 0.0990575999021530...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,651
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
20
null
null
20
548
0.091082
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.129951
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.1299513578414917, 0.12803009152412415, 0.1268633008003235, 0.12653879821300507, 0.12435273081064224, 0.11855022609233856, 0.11546293646097183, 0.11259667575359344, 0.11109207570552826, 0.1086130440235138, 0.10709623247385025, 0.1016058474779129, 0.10097184777259827, 0.10065925121307373, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,652
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
60
null
null
24
548
0.100618
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.132651
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1CC(CO1)C2=NC(=C...
[ 0.13265091180801392, 0.13003598153591156, 0.1263757348060608, 0.12617401778697968, 0.12411369383335114, 0.12080752849578857, 0.12074874341487885, 0.1204552873969078, 0.11911328136920929, 0.11859499663114548, 0.11699309945106506, 0.11617232859134674, 0.11494778096675873, 0.1079593300819397,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,653
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
30
null
null
23
548
0.094252
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.127789
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.1277889907360077, 0.1272742599248886, 0.12480823695659637, 0.12415825575590134, 0.12191653251647949, 0.11692950874567032, 0.11142688989639282, 0.10874026268720627, 0.10799054801464081, 0.10471339523792267, 0.10437463223934174, 0.10359072685241699, 0.10260002315044403, 0.09920788556337357...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,654
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M-H]-
null
null
264.04892
20
null
null
20
548
0.090819
C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O
0.130064
[ "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.13006432354450226, 0.12820905447006226, 0.12697987258434296, 0.12672559916973114, 0.12458190321922302, 0.1187700480222702, 0.11569836735725403, 0.11290988326072693, 0.11126941442489624, 0.10881330072879791, 0.10730239748954773, 0.10178110748529434, 0.1009618267416954, 0.10059791058301926...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,655
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
20
null
null
24
548
0.051297
C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F
0.140428
[ "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1CC(CO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CC(OC1)CC2=NC(=C...
[ 0.1404283046722412, 0.13650697469711304, 0.1309310346841812, 0.13066795468330383, 0.12814520299434662, 0.12739521265029907, 0.124916210770607, 0.12195078283548355, 0.12109807133674622, 0.12090889364480972, 0.11982966959476471, 0.11045826971530914, 0.10964322090148926, 0.10920293629169464, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,656
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
20
null
null
23
548
0.039394
C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O
0.120366
[ "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1CC(CO1)C2=NC(=C...
[ 0.12036643922328949, 0.11872557550668716, 0.1078973338007927, 0.10740651190280914, 0.10288181900978088, 0.09837306290864944, 0.09833638370037079, 0.09533707797527313, 0.09222222864627838, 0.09169252961874008, 0.09108045697212219, 0.08359082788228989, 0.08227445930242538, 0.0822568684816360...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,657
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
60
null
null
22
548
0.072946
C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O
0.132909
[ "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.13290922343730927, 0.13214939832687378, 0.1254633367061615, 0.1219758540391922, 0.1214485913515091, 0.11479705572128296, 0.11250311136245728, 0.10847939550876617, 0.10639329254627228, 0.10519745945930481, 0.10342289507389069, 0.09777688980102539, 0.09514356404542923, 0.09499412775039673,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,658
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
30
null
null
23
548
0.037644
C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O
0.129456
[ "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.1294555813074112, 0.12173032760620117, 0.1122504472732544, 0.11221375316381454, 0.10701967030763626, 0.1028287336230278, 0.0979938805103302, 0.09614872187376022, 0.09361602365970612, 0.0932052731513977, 0.09313833713531494, 0.0860745832324028, 0.08593577891588211, 0.0838177502155304, 0...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,659
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
20
null
null
23
548
0.026243
C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O
0.118728
[ "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.11872812360525131, 0.11164641380310059, 0.1013985425233841, 0.10060727596282959, 0.09482180327177048, 0.09186197817325592, 0.08666907250881195, 0.08458684384822845, 0.08198146522045135, 0.08171135932207108, 0.08138248324394226, 0.0750221461057663, 0.07449637353420258, 0.07294315099716187...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,660
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
60
null
null
22
548
0.072569
C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O
0.132246
[ "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.13224615156650543, 0.13128769397735596, 0.124507836997509, 0.12099616229534149, 0.1204427033662796, 0.1138584092259407, 0.11124256998300552, 0.1072225570678711, 0.10515188425779343, 0.10392694175243378, 0.10218553990125656, 0.09664690494537354, 0.09397776424884796, 0.09385134279727936, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,661
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
30
null
null
23
548
0.037591
C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O
0.129509
[ "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.12950897216796875, 0.1217559352517128, 0.11228005588054657, 0.1122361570596695, 0.10704909265041351, 0.10286904871463776, 0.09801138937473297, 0.09617774933576584, 0.09364242851734161, 0.09322348237037659, 0.09316875785589218, 0.08611610531806946, 0.08598088473081589, 0.08385583758354187...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,662
test
CC(O)(Cn1cc(C(F)(F)F)ccc1=O)C(=O)O
[M+H]+
null
null
266.06347
20
null
null
23
548
0.026201
C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O
0.118772
[ "C1CC2(CN(CC2C1=O)C(=O)C(F)(F)F)C(=O)O", "C1CN(C2C(C1=O)CC2C(=O)O)C(=O)C(F)(F)F", "C1COCCC1C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CC1C2=C(OC(=N2)COCC(F)(F)F)C(=O)O", "C1CC(COC1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "C1CCOC(C1)C2=C(OC(=N2)C(F)(F)F)C(=O)O", "CC1C(CCO1)C2=NC(=C(O2)C(=O)O)C(F)(F)F", "CC1CC(CO1)C2=NC(=C...
[ 0.118772491812706, 0.11170276999473572, 0.10145841538906097, 0.10066082328557968, 0.09488575905561447, 0.09193804860115051, 0.08674400299787521, 0.08467280864715576, 0.08205921947956085, 0.08177777379751205, 0.08145289123058319, 0.07511002570390701, 0.07458490878343582, 0.07303528487682343...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,663
test
CN(CC(=O)O)S(=O)(=O)c1ccc(C(F)(F)F)cc1
[M-H]-
null
null
296.02099
20
null
null
40
369
0.071233
C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N
0.129755
[ "C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N", "C1CC2=NC(C=CC2C(=O)C1)OS(=O)(=O)C(F)(F)F", "C1COC2=C1C=C(C=C2)S(=O)(=O)NOCC(F)(F)F", "CC1=C(C=C2CCCN2C1=O)OS(=O)(=O)C(F)(F)F", "CN1C=C(C2=C1CCCC2=O)OS(=O)(=O)C(F)(F)F", "C1CC2N(C(CS2)C(=O)O)C(=O)C1C(=O)C(F)(F)F", "C1C(CN1S(=O)(=O)C2=CC=CC=C2OC(F)(F)F)O", ...
[ 0.12975504994392395, 0.12182135134935379, 0.12180556356906891, 0.11654271185398102, 0.11457385122776031, 0.11398626118898392, 0.11136303097009659, 0.1101251170039177, 0.10955481976270676, 0.10925119370222092, 0.10747916251420975, 0.10523680597543716, 0.10456685721874237, 0.1039305701851844...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,664
test
CN(CC(=O)O)S(=O)(=O)c1ccc(C(F)(F)F)cc1
[M-H]-
null
null
296.02099
20
null
null
40
369
0.065691
C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N
0.119495
[ "C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N", "C1COC2=C1C=C(C=C2)S(=O)(=O)NOCC(F)(F)F", "C1CC2=NC(C=CC2C(=O)C1)OS(=O)(=O)C(F)(F)F", "CC1=C(C=C2CCCN2C1=O)OS(=O)(=O)C(F)(F)F", "CN1C=C(C2=C1CCCC2=O)OS(=O)(=O)C(F)(F)F", "C1CC2N(C(CS2)C(=O)O)C(=O)C1C(=O)C(F)(F)F", "C1C(CN1S(=O)(=O)C2=CC=CC=C2OC(F)(F)F)O", ...
[ 0.11949493736028671, 0.11320105195045471, 0.1108282282948494, 0.10774131119251251, 0.10438112914562225, 0.10358600318431854, 0.10191451013088226, 0.0991186574101448, 0.09887083619832993, 0.09885774552822113, 0.09704003483057022, 0.09628555923700333, 0.09383081644773483, 0.09323256462812424...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,665
test
CN(CC(=O)O)S(=O)(=O)c1ccc(C(F)(F)F)cc1
[M-H]-
null
null
296.02099
60
null
null
40
369
0.069562
C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N
0.124756
[ "C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N", "C1CC2N(C(CS2)C(=O)O)C(=O)C1C(=O)C(F)(F)F", "CN1C=C(C2=C1CCCC2=O)OS(=O)(=O)C(F)(F)F", "C1CC2=NC(C=CC2C(=O)C1)OS(=O)(=O)C(F)(F)F", "C1COC2=C1C=C(C=C2)S(=O)(=O)NOCC(F)(F)F", "C1C(CN1C(=O)C(F)(F)F)S(=O)(=O)CC2=CC=CO2", "C1C(CN1S(=O)(=O)C2=CC=CC=C2OC(F)(F)F)O", ...
[ 0.12475603073835373, 0.1217767521739006, 0.12127978354692459, 0.12002746015787125, 0.11764505505561829, 0.11652063578367233, 0.1162724569439888, 0.11402042210102081, 0.1132298931479454, 0.11308586597442627, 0.11218518763780594, 0.1082913875579834, 0.10663069784641266, 0.10607846081256866, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,666
test
CN(CC(=O)O)S(=O)(=O)c1ccc(C(F)(F)F)cc1
[M-H]-
null
null
296.02099
30
null
null
39
369
0.067032
C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N
0.115261
[ "C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N", "C1COC2=C1C=C(C=C2)S(=O)(=O)NOCC(F)(F)F", "C1CC2=NC(C=CC2C(=O)C1)OS(=O)(=O)C(F)(F)F", "CC1=C(C=C2CCCN2C1=O)OS(=O)(=O)C(F)(F)F", "CN1C=C(C2=C1CCCC2=O)OS(=O)(=O)C(F)(F)F", "C1C(CN1S(=O)(=O)C2=CC=CC=C2OC(F)(F)F)O", "C1CC2=C(C=CC(N2)OS(=O)(=O)C(F)(F)F)C(=O)C1", ...
[ 0.1152612566947937, 0.11011625081300735, 0.10637794435024261, 0.1032266616821289, 0.09802182763814926, 0.09658533334732056, 0.09604749083518982, 0.09576127678155899, 0.09546038508415222, 0.093816839158535, 0.09300344437360764, 0.09054569154977798, 0.08823060244321823, 0.0876014456152916, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,667
test
CN(CC(=O)O)S(=O)(=O)c1ccc(C(F)(F)F)cc1
[M-H]-
null
null
296.02099
20
null
null
41
369
0.060966
C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N
0.107966
[ "C1COC2=C(O1)C=CC(=C2)C(C(F)(F)F)S(=O)(=O)N", "C1COC2=C1C=C(C=C2)S(=O)(=O)NOCC(F)(F)F", "C1CC2=NC(C=CC2C(=O)C1)OS(=O)(=O)C(F)(F)F", "CC1=C(C=C2CCCN2C1=O)OS(=O)(=O)C(F)(F)F", "CN1C=C(C2=C1CCCC2=O)OS(=O)(=O)C(F)(F)F", "C1C2=CC=CC=C2NC1=O.C(C(F)(F)F)S(=O)(=O)O", "C1C(CN1S(=O)(=O)C2=CC=CC=C2OC(F)(F)F)O", ...
[ 0.10796581953763962, 0.10391323268413544, 0.09882224351167679, 0.09819545596837997, 0.09007192403078079, 0.08911430835723877, 0.08899878710508347, 0.08876969665288925, 0.08741848170757294, 0.08482569456100464, 0.08384175598621368, 0.08230946213006973, 0.08214104920625687, 0.079366914927959...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,668
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
20
null
null
544
4,603
0.125738
C1=CNC(Oc2ccccn2)C=C1
0.152109
[ "C1=CNC(Oc2ccccn2)C=C1", "NNc1ccc2ccc(O)cc2c1", "Cc1ccc2c(c1)=NCC(=O)CN=2", "O=NCCc1cc2ccccc2[nH]1", "N#Cc1ccn(CC2CC2)c(=O)c1", "C#C.CNc1nc2ccccc2o1", "N#CN1CCc2c(O)cccc2C1", "OCCc1ccc2nccnc2c1", "OCCc1ccc2ncncc2c1", "N#CC1(C(=O)c2ccc[nH]2)CCC1", "NC1=CC=C(c2ccccn2)OC1", "CC(N=O)c1cc2ccccc2[nH...
[ 0.15210866928100586, 0.14800916612148285, 0.14731159806251526, 0.14699679613113403, 0.14690029621124268, 0.14622938632965088, 0.14567619562149048, 0.14567604660987854, 0.1456625759601593, 0.14550793170928955, 0.14542452991008759, 0.14524626731872559, 0.14506348967552185, 0.1443700492382049...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,669
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
20
null
null
858
4,603
0.106012
OCCc1ccc2nccnc2c1
0.147503
[ "OCCc1ccc2nccnc2c1", "NNc1cc(O)c2ccccc2c1", "NCOc1ccc2ncccc2c1", "NOCc1ccc2ncccc2c1", "NOCc1ccc2ccncc2c1", "OCCc1ccc2ncncc2c1", "NOCc1ccc2cnccc2c1", "NNc1ccc2ccc(O)cc2c1", "NOCc1ccc2cccnc2c1", "CONc1ccc2ncccc2c1", "NC1=CC=C(c2ccccn2)OC1", "OCCc1ccc2cnncc2c1", "Cc1ccc2ncccc2c1.N=O", "C1=CNC...
[ 0.14750255644321442, 0.1460709571838379, 0.14444959163665771, 0.14410549402236938, 0.14388282597064972, 0.14365561306476593, 0.14309272170066833, 0.14249813556671143, 0.14132530987262726, 0.13901104032993317, 0.137356698513031, 0.13654009997844696, 0.1358419805765152, 0.13324551284313202, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,670
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
60
null
null
3,932
4,603
0.083053
Nc1ccccc1Nc1ccco1
0.167247
[ "Nc1ccccc1Nc1ccco1", "Nc1ccc(Nc2ccco2)cc1", "Nc1cc(Cc2ccoc2)ccn1", "NCOc1ccc2ncccc2c1", "Oc1ccc(Nn2cccc2)cc1", "CONc1ccc2ncccc2c1", "Nc1cc(Cc2ccco2)ccn1", "Oc1cccc(Nn2cccc2)c1", "NCOc1ccc2cccnc2c1", "N#Cc1ccc2c(c1)OCCNC2", "N#Cc1cccc(OC2CCC2)n1", "Oc1ccccc1.c1cncnc1", "N#CN(c1ccccc1)C1COC1",...
[ 0.1672469675540924, 0.16606667637825012, 0.1640780121088028, 0.1634986400604248, 0.16033005714416504, 0.15992864966392517, 0.15726691484451294, 0.156910240650177, 0.1567554473876953, 0.1555207371711731, 0.15512940287590027, 0.15507060289382935, 0.15488609671592712, 0.15447139739990234, 0...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,671
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
20
null
null
682
4,603
0.088756
NOCc1ccc2cnccc2c1
0.124755
[ "NOCc1ccc2cnccc2c1", "OCCc1ccc2nccnc2c1", "NOCc1ccc2ncccc2c1", "COc1ccc2nccnc2c1C", "NCOc1ccc2ncccc2c1", "O=CCCc1ccc2cn[nH]c2c1", "NOCc1ccc2ccncc2c1", "NOCc1ccc2cccnc2c1", "CCOc1ccc2nccnc2c1", "NOCc1ccc2ccccc2n1", "O=CCCc1ccc2nc[nH]c2c1", "O=c1[nH]c2ccccc2n1C1CC1", "O=NCCc1cc2ccccc2[nH]1", ...
[ 0.1247551292181015, 0.12393363565206528, 0.12339600175619125, 0.12318751215934753, 0.1230400800704956, 0.12253764271736145, 0.12236963957548141, 0.12227875739336014, 0.12206301838159561, 0.12172012776136398, 0.1211901307106018, 0.12093637138605118, 0.12018152326345444, 0.11952142417430878,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,672
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
45
null
null
2,643
4,603
0.125108
N#Cc1ccccc1NC1COC1
0.17966
[ "N#Cc1ccccc1NC1COC1", "N#CN(c1ccccc1)C1COC1", "N#Cc1ccc2c(c1)OCCNC2", "N#Cc1ccccc1OC1CNC1", "OCC#Cc1ccc(C2CC2)nn1", "N#Cc1ncccc1OC1CCC1", "N#Cc1cccc(OC2CCC2)n1", "N#Cc1cc(N)ccc1OC1CC1", "N#Cc1cccc(NC2COC2)c1", "N#Cc1ccc(N)cc1OC1CC1", "N#Cc1cccc(OCC2CC2)n1", "N#Cc1ccc(NCC2CO2)cc1", "N#CN1CCc2...
[ 0.17966020107269287, 0.1787944734096527, 0.17858803272247314, 0.177700012922287, 0.1775091588497162, 0.17724108695983887, 0.17625001072883606, 0.1760421097278595, 0.17603498697280884, 0.1756420135498047, 0.17558148503303528, 0.17543864250183105, 0.17535322904586792, 0.17487740516662598, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,673
test
NC(=O)Cc1c[nH]c2ccccc12
[M+H]+
null
null
175.08659
15
null
null
957
4,603
0.093692
Cc1cc2[nH]ccc(=O)c2nc1C
0.129992
[ "Cc1cc2[nH]ccc(=O)c2nc1C", "Cc1cc2c(ccc(=O)n2C)cn1", "Cc1nc2ccccn2c(=O)c1C", "Cc1cc2ccncc2n(C)c1=O", "Cc1ccc2nc(C)cc(=O)n2c1", "C=C1c2ccccc2C(=O)NN1C", "Cc1cnc2ccn(C)c(=O)c2c1", "Cc1cc2ccncc2c(=O)n1C", "Cc1cc2cnccc2n(C)c1=O", "Cc1ccc2cnn(C)c(=O)c2c1", "Cc1cccc2c1ncc(=O)n2C", "Cc1cc2cccnc2n(C)c...
[ 0.12999199330806732, 0.12952443957328796, 0.12906503677368164, 0.12799786031246185, 0.12766170501708984, 0.12709112465381622, 0.12599588930606842, 0.1255817413330078, 0.1254345327615738, 0.12434536963701248, 0.12357570230960846, 0.12338000535964966, 0.1232171505689621, 0.12319648265838623,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,674
test
NC(=O)Cc1c[nH]c2ccccc12
[M+H]+
null
null
175.08659
15
null
null
758
4,603
0.073636
Cc1cc2ccncc2n(C)c1=O
0.104999
[ "Cc1cc2ccncc2n(C)c1=O", "Cc1cc2[nH]ccc(=O)c2nc1C", "Cc1nc2cc3c(cc2[nH]1)CCO3", "Cc1[nH]c(=O)nc2c1C=CCC=C2", "Cc1ccc2nc(C)cc(=O)n2c1", "Cc1nc2cc3c(cc2[nH]1)COC3", "Cc1cnc2[nH]c(=O)c(C)cc2c1", "Cc1cc2cnccc2n(C)c1=O", "C=CC(O)c1nc2ccccc2[nH]1", "Cc1cnc2ccn(C)c(=O)c2c1", "Cc1ccc2[nH]c(=O)cnc2c1C", ...
[ 0.10499872267246246, 0.10358203947544098, 0.10345876216888428, 0.10299859941005707, 0.10269448906183243, 0.10234186798334122, 0.10198665410280228, 0.10190193355083466, 0.10161297023296356, 0.10116887092590332, 0.1002492904663086, 0.10013248026371002, 0.09999115020036697, 0.0999900624155998...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,675
test
NC(=O)Cc1c[nH]c2ccccc12
[M+H]+
null
null
175.08659
60
null
null
624
4,603
0.081865
Cc1cc2[nH]ccc(=O)c2nc1C
0.109898
[ "Cc1cc2[nH]ccc(=O)c2nc1C", "Cc1cc2ccncc2n(C)c1=O", "Cc1ccc2nc(C)cc(=O)n2c1", "C=CC(O)c1nc2ccccc2[nH]1", "Cc1[nH]c(=O)nc2c1C=CCC=C2", "Cc1cc2c(ccc(=O)n2C)cn1", "Cc1cnc2ccn(C)c(=O)c2c1", "C=C1c2ccccc2C(=O)NN1C", "Cc1cc2cnccc2n(C)c1=O", "Cc1cnc2[nH]c(=O)c(C)cc2c1", "Cc1nc2cc3c(cc2[nH]1)CCO3", "CC...
[ 0.10989787429571152, 0.1093103215098381, 0.10853137820959091, 0.10767923295497894, 0.10664598643779755, 0.10636427998542786, 0.10618283599615097, 0.10595853626728058, 0.10594692081212997, 0.10582706332206726, 0.1052529439330101, 0.10518648475408554, 0.10516466200351715, 0.10506176948547363...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,676
test
NC(=O)Cc1c[nH]c2ccccc12
[M+H]+
null
null
175.08659
20
null
null
550
4,603
0.064574
C=CC(O)c1nc2ccccc2[nH]1
0.091013
[ "C=CC(O)c1nc2ccccc2[nH]1", "Cc1cnc2[nH]c(=O)c(C)cc2c1", "Cc1cc2ccncc2n(C)c1=O", "CC=C(C#CC(=O)C#N)C=C(C)N", "Cc1nc2cc(C=O)c(C)cc2[nH]1", "Cc1cc2[nH]ccc(=O)c2nc1C", "Cc1nc2c(C=O)c(C)ccc2[nH]1", "Cc1ccc2[nH]c(=O)cnc2c1C", "Cc1ccc2nc(C)cc(=O)n2c1", "CCc1cc2[nH]c(=O)ccc2cn1", "Cc1cc2[nH]c(=O)ccc2c(C...
[ 0.09101313352584839, 0.09005186706781387, 0.08943416178226471, 0.08916787058115005, 0.08802960067987442, 0.08755747228860855, 0.08713644742965698, 0.08703496307134628, 0.08682359755039215, 0.08595944195985794, 0.08591176569461823, 0.0855022594332695, 0.0853225588798523, 0.08513493835926056...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,677
test
NC(=O)Cc1c[nH]c2ccccc12
[M+H]+
null
null
175.08659
15
null
null
583
4,603
0.062415
C=CC(O)c1nc2ccccc2[nH]1
0.088864
[ "C=CC(O)c1nc2ccccc2[nH]1", "Cc1cnc2[nH]c(=O)c(C)cc2c1", "Cc1cc2ccncc2n(C)c1=O", "CC=C(C#CC(=O)C#N)C=C(C)N", "Cc1nc2cc(C=O)c(C)cc2[nH]1", "Cc1cc2[nH]ccc(=O)c2nc1C", "Cc1nc2c(C=O)c(C)ccc2[nH]1", "Cc1ccc2[nH]c(=O)cnc2c1C", "Cc1ccc2nc(C)cc(=O)n2c1", "Cc1nc2cc3c(cc2[nH]1)CCO3", "Cc1cc2[nH]c(=O)ccc2c(...
[ 0.08886449038982391, 0.0885612964630127, 0.08820299804210663, 0.0870567336678505, 0.0864512175321579, 0.08579687029123306, 0.08550727367401123, 0.08547760546207428, 0.08513946831226349, 0.08490585535764694, 0.08470426499843597, 0.08445438742637634, 0.08423259109258652, 0.08372921496629715,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,678
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
45
null
null
172
4,603
0.093419
C1=CNc2nc3c(cc2C1)OCC3
0.132539
[ "C1=CNc2nc3c(cc2C1)OCC3", "c1cc2c(cn1)OCC1=C2CCN1", "Cc1nc2n(c1C=O)C=CCC=C2", "C1=CC2=C(C=CC3CCN=C23)NO1", "C1=Cc2c(ccc3c2NCC3)NO1", "c1ncc2c3c(oc2n1)CCCC3", "OC1(c2ccccn2)C=CC=CN1", "C1=NN2COc3ccccc3C2C1", "Cc1[nH]c2ccccc2c1C1NO1", "C1=NN2c3ccccc3COC2C1", "Cc1nc2c(c(=O)[nH]1)C=CCC=C2", "Cc1cc...
[ 0.13253924250602722, 0.1234053298830986, 0.12193065136671066, 0.12115345150232315, 0.12001741677522659, 0.11866290122270584, 0.11827483028173447, 0.11807335913181305, 0.11777018010616302, 0.11691446602344513, 0.1165311336517334, 0.1161881685256958, 0.11561429500579834, 0.11507955193519592,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,679
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
45
null
null
181
4,603
0.097962
C1=CNc2nc3c(cc2C1)OCC3
0.140215
[ "C1=CNc2nc3c(cc2C1)OCC3", "C1=Cc2c(ccc3c2NCC3)NO1", "c1cc2c(cn1)OCC1=C2CCN1", "Cc1[nH]c2ccccc2c1C1NO1", "C1=NN2COc3ccccc3C2C1", "C1=CC2=C(C=CC3CCN=C23)NO1", "C1=NN2c3ccccc3COC2C1", "OC1(c2ccccn2)C=CC=CN1", "Cc1nc2n(c1C=O)C=CCC=C2", "OC1(c2cnccn2)C=CC=CC1", "c1ncc2c3c(oc2n1)CCCC3", "Cc1cc2c(o1)...
[ 0.14021465182304382, 0.13365478813648224, 0.1318260133266449, 0.13079431653022766, 0.12993386387825012, 0.1284678876399994, 0.1278604418039322, 0.12696541845798492, 0.12396722286939621, 0.1233895793557167, 0.12215913087129593, 0.122146375477314, 0.12098109722137451, 0.12064076960086823, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,680
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
20
null
null
188
4,603
0.063652
ON1CCc2ccc3[nH]ccc3c21
0.096017
[ "ON1CCc2ccc3[nH]ccc3c21", "NC(=O)c1cc2ccccc2cn1.[HH]", "C=C1c2ccccc2NC(=O)N1C", "CN1C(=O)C2NCc3cccc1c32", "C1=NOC2NCc3ccccc3C12", "C1=NN2c3ccccc3COC2C1", "Cc1c(C=O)n(C)c2ncccc12", "COc1nc2ncccc2cc1C", "OC1(c2ccccn2)C=CC=CN1", "OC1=CCN2c3ccccc3NC12", "O=C1NCc2ccc3c(c21)CCN3", "O=C1CC2CNc3ccccc3...
[ 0.09601747244596481, 0.0934559628367424, 0.08921004086732864, 0.08867906033992767, 0.08806405961513519, 0.08760912716388702, 0.08737985044717789, 0.0865909680724144, 0.08639632165431976, 0.08629152923822403, 0.08619312942028046, 0.08618244528770447, 0.08496934920549393, 0.08482867479324341...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,681
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
60
null
null
1,548
4,603
0.097531
CNc1cc(O)c2ncccc2c1
0.148715
[ "CNc1cc(O)c2ncccc2c1", "NCc1cc(O)c2cnccc2c1", "NCc1cc(O)c2ncccc2c1", "COc1cc(N)c2ccncc2c1", "NCc1cc(O)c2cccnc2c1", "COc1cc(N)c2ncccc2c1", "Cc1cc2cc(O)ccc2c(N)n1", "Cc1cc(C#N)c2c(c1)OCCN2", "Cc1cc(N)c2ccc(O)cc2n1", "Cc1cc2ccccc2n1C(N)=O", "COc1cc(N)c2cccnc2c1", "Cc1cnc2cc(O)c(N)cc2c1", "N#Cc1...
[ 0.1487150937318802, 0.14448410272598267, 0.14313143491744995, 0.14306855201721191, 0.14132115244865417, 0.14079973101615906, 0.1402527242898941, 0.13977673649787903, 0.13881614804267883, 0.1370786726474762, 0.13670200109481812, 0.13667765259742737, 0.13606613874435425, 0.13522765040397644,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,682
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
45
null
null
479
4,603
0.11519
Cc1cc2ccncc2n(C)c1=O
0.14095
[ "Cc1cc2ccncc2n(C)c1=O", "Cc1cc2cnccc2n(C)c1=O", "Cc1ccc2cnn(C)c(=O)c2c1", "Cc1cnc2ccn(C)c(=O)c2c1", "Cc1cc2cccnc2n(C)c1=O", "CNc1cc(O)c2ncccc2c1", "Cc1cc(C=O)c2c(cnn2C)c1", "Cc1cc(N)c2ccc(O)cc2n1", "C=C1c2ccccc2C(=O)NN1C", "Cc1ccc2ncn(C)c(=O)c2c1", "Cc1cc2c(ccc(=O)n2C)cn1", "Cc1cc2[nH]ccc(=O)c...
[ 0.1409500539302826, 0.14006684720516205, 0.13533790409564972, 0.13444088399410248, 0.13436606526374817, 0.1332980841398239, 0.1325170248746872, 0.13168074190616608, 0.13135357201099396, 0.13127362728118896, 0.13119657337665558, 0.13097292184829712, 0.1309293508529663, 0.13078078627586365, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,683
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
20
null
null
421
4,603
0.124742
O=NCCc1cc2ccccc2[nH]1
0.14801
[ "O=NCCc1cc2ccccc2[nH]1", "C1=CNC(Oc2ccccn2)C=C1", "C#C.CNc1nc2ccccc2o1", "CC(N=O)c1cc2ccccc2[nH]1", "N#CC1(C(=O)c2ccc[nH]2)CCC1", "N#Cc1ccn(CC2CC2)c(=O)c1", "NNc1ccc2ccc(O)cc2c1", "CON=Cc1ccc2cc[nH]c2c1", "NC1=CC=C(c2ccccn2)OC1", "N#CN1CCc2c(O)cccc2C1", "Cc1ccc2ncccc2c1.N=O", "Cc1ccc2c(c1)=NCC...
[ 0.14800985157489777, 0.14737722277641296, 0.1446993052959442, 0.14376266300678253, 0.14357233047485352, 0.14338462054729462, 0.1428389549255371, 0.14211910963058472, 0.1420155167579651, 0.14123502373695374, 0.14118626713752747, 0.14116615056991577, 0.14111025631427765, 0.14074566960334778,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,684
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
20
null
null
677
4,603
0.107418
OCCc1ccc2nccnc2c1
0.144018
[ "OCCc1ccc2nccnc2c1", "NOCc1ccc2ncccc2c1", "NCOc1ccc2ncccc2c1", "NOCc1ccc2cnccc2c1", "NOCc1ccc2ccncc2c1", "NNc1cc(O)c2ccccc2c1", "OCCc1ccc2ncncc2c1", "NNc1ccc2ccc(O)cc2c1", "NOCc1ccc2cccnc2c1", "Cc1ccc2ncccc2c1.N=O", "NC1=CC=C(c2ccccn2)OC1", "CONc1ccc2ncccc2c1", "CN1C(=O)C2NCc3cccc1c32", "O...
[ 0.1440175324678421, 0.14156368374824524, 0.14123056828975677, 0.14072002470493317, 0.1405605971813202, 0.13993242383003235, 0.13919663429260254, 0.13860684633255005, 0.1384904831647873, 0.13762177526950836, 0.13592195510864258, 0.1357642412185669, 0.1341303586959839, 0.13184404373168945, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,685
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
60
null
null
3,823
4,603
0.092987
Nc1ccc(Nc2ccco2)cc1
0.171321
[ "Nc1ccc(Nc2ccco2)cc1", "Nc1ccccc1Nc1ccco1", "Nc1cc(Cc2ccoc2)ccn1", "NCOc1ccc2ncccc2c1", "Oc1ccc(Nn2cccc2)cc1", "CONc1ccc2ncccc2c1", "N#Cc1ccccc1NC1COC1", "N#CN(c1ccccc1)C1COC1", "N#Cc1cccc(OC2CCC2)n1", "N#Cc1ccc2c(c1)OCCNC2", "Nc1cc(Cc2ccco2)ccn1", "Oc1cccc(Nn2cccc2)c1", "N#Cc1ccncc1OC1CCC1"...
[ 0.17132097482681274, 0.17049908638000488, 0.16923455893993378, 0.16836270689964294, 0.1672951728105545, 0.16470974683761597, 0.16383931040763855, 0.1637476086616516, 0.1634855717420578, 0.16341528296470642, 0.16316819190979004, 0.16307465732097626, 0.16143137216567993, 0.161196768283844, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,686
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
20
null
null
610
4,603
0.090328
COc1ccc2nccnc2c1C
0.124657
[ "COc1ccc2nccnc2c1C", "O=CCCc1ccc2cn[nH]c2c1", "NOCc1ccc2cnccc2c1", "OCCc1ccc2nccnc2c1", "O=CCCc1ccc2nc[nH]c2c1", "CCOc1ccc2nccnc2c1", "Cc1ccc2ncccc2c1.N=O", "O=c1[nH]c2ccccc2n1C1CC1", "NOCc1ccc2ncccc2c1", "NCOc1ccc2ncccc2c1", "O=NCCc1cc2ccccc2[nH]1", "NOCc1ccc2ccncc2c1", "NOCc1ccc2cccnc2c1",...
[ 0.12465721368789673, 0.1239662915468216, 0.12338536977767944, 0.12322544306516647, 0.12284234911203384, 0.12270936369895935, 0.12268643826246262, 0.12258081883192062, 0.12241023033857346, 0.12156596779823303, 0.12120705842971802, 0.12103244662284851, 0.1206289678812027, 0.12050001323223114...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,687
test
CC1=NN(c2ccccc2)C(=O)C1
[M-H]-
null
null
173.07204
45
null
null
2,538
4,603
0.124173
N#Cc1ccccc1NC1COC1
0.178396
[ "N#Cc1ccccc1NC1COC1", "N#CN(c1ccccc1)C1COC1", "N#Cc1ncccc1OC1CCC1", "N#Cc1cc(N)ccc1OC1CC1", "N#Cc1ccccc1OC1CNC1", "N#Cc1ccc(N)cc1OC1CC1", "OCC#Cc1ccc(C2CC2)nn1", "N#Cc1ccc2c(c1)OCCNC2", "N#CN1CCc2c(O)cccc2C1", "N#Cc1cccc(NC2COC2)c1", "N#Cc1ccncc1OC1CCC1", "N#CN1CCOc2ccccc2C1", "N#Cc1cccc(OC2...
[ 0.17839618027210236, 0.17742738127708435, 0.1767403930425644, 0.17668692767620087, 0.1764775812625885, 0.17530858516693115, 0.17463469505310059, 0.17444315552711487, 0.17418614029884338, 0.17418044805526733, 0.17408844828605652, 0.17402240633964539, 0.17397168278694153, 0.17393633723258972...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,688
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
20
null
null
191
4,603
0.093459
C1=CNc2nc3c(cc2C1)OCC3
0.135256
[ "C1=CNc2nc3c(cc2C1)OCC3", "c1cc2c(cn1)OCC1=C2CCN1", "C1=CC2=C(C=CC3CCN=C23)NO1", "C1=Cc2c(ccc3c2NCC3)NO1", "Cc1nc2n(c1C=O)C=CCC=C2", "Cc1[nH]c2ccccc2c1C1NO1", "C1=NN2COc3ccccc3C2C1", "OC1(c2ccccn2)C=CC=CN1", "c1ncc2c3c(oc2n1)CCCC3", "C1=NN2c3ccccc3COC2C1", "Cc1nc2c(c(=O)[nH]1)C=CCC=C2", "Cc1cc...
[ 0.13525602221488953, 0.1275826394557953, 0.12417525053024292, 0.12370441854000092, 0.12253846973180771, 0.12134012579917908, 0.12067350000143051, 0.12026495486497879, 0.12008883059024811, 0.11903470009565353, 0.1174486055970192, 0.11694074422121048, 0.11620517820119858, 0.11593283712863922...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,689
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
20
null
null
193
4,603
0.09884
C1=CNc2nc3c(cc2C1)OCC3
0.142776
[ "C1=CNc2nc3c(cc2C1)OCC3", "C1=Cc2c(ccc3c2NCC3)NO1", "c1cc2c(cn1)OCC1=C2CCN1", "Cc1[nH]c2ccccc2c1C1NO1", "C1=NN2COc3ccccc3C2C1", "C1=CC2=C(C=CC3CCN=C23)NO1", "OC1(c2ccccn2)C=CC=CN1", "C1=NN2c3ccccc3COC2C1", "OC1(c2cnccn2)C=CC=CC1", "Cc1nc2n(c1C=O)C=CCC=C2", "Cc1cc2c(o1)CCc1cn[nH]c1-2", "c1ccc2c...
[ 0.14277571439743042, 0.13565212488174438, 0.13514471054077148, 0.13275891542434692, 0.131877601146698, 0.13081204891204834, 0.12979847192764282, 0.12977370619773865, 0.12581117451190948, 0.12563960254192352, 0.1246732771396637, 0.12439661473035812, 0.12407559156417847, 0.12342493236064911,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,690
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
60
null
null
2,260
4,603
0.081986
N#Cc1ccc2c(c1)OCCCN2
0.143645
[ "N#Cc1ccc2c(c1)OCCCN2", "CNc1cc(O)c2ncccc2c1", "N#Cc1ccc2c(c1)NCCCO2", "NCc1cc(O)c2cnccc2c1", "Cc1cc(C#N)c2c(c1)OCCN2", "NCc1cc(O)c2ncccc2c1", "NCc1cc(O)c2cccnc2c1", "N#Cc1ccc2c(c1)OCCNC2", "N#Cc1cccc2c1OCCCN2", "OCC#Cc1ccc(C2CC2)nn1", "N#CCc1ccc2c(c1)OCCN2", "N#Cc1ccc2c(n1)CCCC2O", "N#Cc1cc...
[ 0.1436445564031601, 0.14100106060504913, 0.1402912437915802, 0.13991814851760864, 0.1391610950231552, 0.13858827948570251, 0.13822732865810394, 0.13797827064990997, 0.1373061239719391, 0.13433989882469177, 0.13373249769210815, 0.1330775022506714, 0.13302139937877655, 0.13277116417884827, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,691
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
20
null
null
197
4,603
0.063696
ON1CCc2ccc3[nH]ccc3c21
0.097086
[ "ON1CCc2ccc3[nH]ccc3c21", "NC(=O)c1cc2ccccc2cn1.[HH]", "CN1C(=O)C2NCc3cccc1c32", "C=C1c2ccccc2NC(=O)N1C", "C1=NOC2NCc3ccccc3C12", "Cc1c(C=O)n(C)c2ncccc12", "C1=NN2c3ccccc3COC2C1", "COc1nc2ncccc2cc1C", "OC1(c2ccccn2)C=CC=CN1", "O=C1CC2CNc3ccccc3N12", "O=C1NCc2ccc3c(c21)CCN3", "OC1=CCN2c3ccccc3N...
[ 0.09708566963672638, 0.09471279382705688, 0.08953029662370682, 0.08939826488494873, 0.08829724788665771, 0.08796457946300507, 0.08762487769126892, 0.08694624155759811, 0.08652941882610321, 0.0864892229437828, 0.0864114761352539, 0.08638590574264526, 0.08604668825864792, 0.08539728820323944...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,692
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
45
null
null
695
4,603
0.115521
Cc1cc2ccncc2n(C)c1=O
0.145715
[ "Cc1cc2ccncc2n(C)c1=O", "Cc1cc2cnccc2n(C)c1=O", "CNc1cc(O)c2ncccc2c1", "Cc1cc(N)c2ccc(O)cc2n1", "COc1cc(N)c2ccncc2c1", "Cc1ccc2cnn(C)c(=O)c2c1", "Cc1cc2cccnc2n(C)c1=O", "Cc1cc2ccncc2c(=O)n1C", "Cc1cc(C=O)c2c(cnn2C)c1", "Cc1cc(N)c2cc(O)ccc2n1", "CC(=O)Cc1cc2cc[nH]c2cn1", "Cc1cnc2ccn(C)c(=O)c2c1...
[ 0.1457151472568512, 0.14546912908554077, 0.1438325196504593, 0.1408987045288086, 0.1399608552455902, 0.1395615041255951, 0.13920526206493378, 0.1377403438091278, 0.13764743506908417, 0.1373736560344696, 0.13722842931747437, 0.13718891143798828, 0.13678336143493652, 0.1366642564535141, 0....
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,693
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
60
null
null
2,256
4,603
0.08135
N#Cc1ccc2c(c1)OCCCN2
0.14316
[ "N#Cc1ccc2c(c1)OCCCN2", "CNc1cc(O)c2ncccc2c1", "N#Cc1ccc2c(c1)NCCCO2", "NCc1cc(O)c2cnccc2c1", "Cc1cc(C#N)c2c(c1)OCCN2", "NCc1cc(O)c2ncccc2c1", "NCc1cc(O)c2cccnc2c1", "N#Cc1ccc2c(c1)OCCNC2", "N#Cc1cccc2c1OCCCN2", "OCC#Cc1ccc(C2CC2)nn1", "N#CCc1ccc2c(c1)OCCN2", "N#Cc1ccc(N)c(OC2CC2)c1", "N#Cc1...
[ 0.1431596577167511, 0.14044570922851562, 0.13964048027992249, 0.13944733142852783, 0.13876256346702576, 0.13812199234962463, 0.13777905702590942, 0.13724324107170105, 0.13668666779994965, 0.1336270570755005, 0.13307921588420868, 0.13261821866035461, 0.13248521089553833, 0.1322748214006424,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,694
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
20
null
null
197
4,603
0.062759
ON1CCc2ccc3[nH]ccc3c21
0.096798
[ "ON1CCc2ccc3[nH]ccc3c21", "NC(=O)c1cc2ccccc2cn1.[HH]", "C=C1c2ccccc2NC(=O)N1C", "CN1C(=O)C2NCc3cccc1c32", "C1=NOC2NCc3ccccc3C12", "Cc1c(C=O)n(C)c2ncccc12", "O=C1CC2CNc3ccccc3N12", "C1=NN2c3ccccc3COC2C1", "O=C1NCc2ccc3c(c21)CCN3", "COc1nc2ncccc2cc1C", "OC1=CCN2c3ccccc3NC12", "NN1C(=O)CC=Cc2cccc...
[ 0.09679801762104034, 0.0939180999994278, 0.08883620798587799, 0.08864246308803558, 0.08760152012109756, 0.08708366751670837, 0.08642301708459854, 0.08640588074922562, 0.0863908976316452, 0.08595578372478485, 0.08592744171619415, 0.08554022014141083, 0.08546444773674011, 0.08533668518066406...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,695
test
CC1=NN(c2ccccc2)C(=O)C1
[M+H]+
null
null
175.08659
45
null
null
693
4,603
0.115285
Cc1cc2ccncc2n(C)c1=O
0.145497
[ "Cc1cc2ccncc2n(C)c1=O", "Cc1cc2cnccc2n(C)c1=O", "CNc1cc(O)c2ncccc2c1", "Cc1cc(N)c2ccc(O)cc2n1", "COc1cc(N)c2ccncc2c1", "Cc1ccc2cnn(C)c(=O)c2c1", "Cc1cc2cccnc2n(C)c1=O", "Cc1cc2ccncc2c(=O)n1C", "Cc1cc(C=O)c2c(cnn2C)c1", "Cc1cc(N)c2cc(O)ccc2n1", "CC(=O)Cc1cc2cc[nH]c2cn1", "Cc1cnc2ccn(C)c(=O)c2c1...
[ 0.1454973816871643, 0.14524106681346893, 0.14358939230442047, 0.14069052040576935, 0.1397225558757782, 0.1394699215888977, 0.13901203870773315, 0.1376093029975891, 0.137490376830101, 0.13711223006248474, 0.13711042702198029, 0.13700523972511292, 0.1366153359413147, 0.13653069734573364, 0...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,696
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
30
null
null
451
4,603
0.142058
O=NCCc1cc2ccccc2[nH]1
0.17627
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "C#C.CNc1nc2ccccc2o1", "OCC=Cc1ccn2ccnc2c1", "N#Cc1ccc(N)cc1OC1CC1", "Cc1cc(C#N)ncc1OC1CC1", "N#Cc1ccc(C=O)n1CC1CC1", "N#Cc1cc(N)ccc1OC1CC1", "N#Cc1ccn(CC2CC2)c(=O)c1", "OCC=Cc1cn2ccccc2n1", "Cc1cnc(C#N)cc1OC1CC1", "O=CCCc1cc2ccncc2[nH]1", "N...
[ 0.1762697696685791, 0.17016032338142395, 0.1692069172859192, 0.16818970441818237, 0.16795380413532257, 0.1671391725540161, 0.1667361557483673, 0.16663596034049988, 0.1656443029642105, 0.16408324241638184, 0.1639811396598816, 0.16392424702644348, 0.1638059914112091, 0.1634466052055359, 0....
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,697
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
30
null
null
757
4,603
0.127629
O=NCCc1cc2ccccc2[nH]1
0.166915
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "C#C.CNc1nc2ccccc2o1", "O=CCCc1ccc2nc[nH]c2c1", "O=CCCc1ccc2cn[nH]c2c1", "N#Cc1ccn(CC2CC2)c(=O)c1", "O=CCCc1cc2ccncc2[nH]1", "N#CC1(C(=O)c2ccc[nH]2)CCC1", "CC(N=O)c1cc2ccccc2[nH]1", "N#Cc1ccc(N)cc1OC1CC1", "O=CCCc1ccc2[nH]ncc2c1", "OCC=Cc1ccc2n...
[ 0.16691471636295319, 0.16020801663398743, 0.15760937333106995, 0.1563909649848938, 0.15497669577598572, 0.15418073534965515, 0.1533803641796112, 0.153377503156662, 0.15213358402252197, 0.15188944339752197, 0.15176397562026978, 0.1509893238544464, 0.15094399452209473, 0.15079990029335022, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,698
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
20
null
null
1,120
4,603
0.116623
O=NCCc1cc2ccccc2[nH]1
0.157921
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "O=CCCc1ccc2nc[nH]c2c1", "O=CCCc1ccc2cn[nH]c2c1", "C#C.CNc1nc2ccccc2o1", "N#CC1(C(=O)c2ccc[nH]2)CCC1", "Cc1ccc2ncccc2c1.N=O", "CC(N=O)c1cc2ccccc2[nH]1", "N#Cc1ccn(CC2CC2)c(=O)c1", "O=CCCc1ccc2[nH]ncc2c1", "O=CCCc1cc2ccncc2[nH]1", "N#CC1(C(=O)c2...
[ 0.15792113542556763, 0.15074191987514496, 0.1497446447610855, 0.1485958844423294, 0.14845307171344757, 0.14624474942684174, 0.14599326252937317, 0.14546337723731995, 0.14488112926483154, 0.1445387750864029, 0.14402548968791962, 0.14297859370708466, 0.14200147986412048, 0.1418634057044983, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,699
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
60
null
null
360
4,603
0.149499
O=NCCc1cc2ccccc2[nH]1
0.185362
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "OCC=Cc1ccn2ccnc2c1", "N#Cc1ccc(C=O)n1CC1CC1", "Cc1cc(C#N)ncc1OC1CC1", "N#Cc1ccc(N)cc1OC1CC1", "N#Cc1cc(N)ccc1OC1CC1", "N#Cc1cccnc1OC1CCC1", "C#C.CNc1nc2ccccc2o1", "N#Cc1ncccc1OC1CCC1", "O=CCCc1cc2ccncc2[nH]1", "OCC=Cc1cn2ccccc2n1", "Cc1cnc(C...
[ 0.1853620409965515, 0.18005695939064026, 0.17737649381160736, 0.1772414743900299, 0.1766192466020584, 0.17626067996025085, 0.17616038024425507, 0.17488732933998108, 0.1738249957561493, 0.17308592796325684, 0.17300328612327576, 0.1725616455078125, 0.17225365340709686, 0.17223194241523743, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,700
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
30
null
null
426
4,603
0.143568
O=NCCc1cc2ccccc2[nH]1
0.176716
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "OCC=Cc1ccn2ccnc2c1", "C#C.CNc1nc2ccccc2o1", "N#Cc1ccc(N)cc1OC1CC1", "N#Cc1ccc(C=O)n1CC1CC1", "N#Cc1cc(N)ccc1OC1CC1", "Cc1cc(C#N)ncc1OC1CC1", "N#Cc1ccn(CC2CC2)c(=O)c1", "OCC=Cc1cn2ccccc2n1", "OCC=Cc1ccc2nc[nH]c2c1", "N#Cc1cccnc1OC1CCC1", "N#C...
[ 0.1767157018184662, 0.1708708256483078, 0.17056594789028168, 0.170124351978302, 0.16841435432434082, 0.16770324110984802, 0.1673640012741089, 0.16726630926132202, 0.16645139455795288, 0.165973961353302, 0.16455432772636414, 0.1643737554550171, 0.16401657462120056, 0.16400016844272614, 0....
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,701
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
45
null
null
363
4,603
0.149929
O=NCCc1cc2ccccc2[nH]1
0.185401
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "OCC=Cc1ccn2ccnc2c1", "N#Cc1ccc(C=O)n1CC1CC1", "Cc1cc(C#N)ncc1OC1CC1", "N#Cc1ccc(N)cc1OC1CC1", "N#Cc1cc(N)ccc1OC1CC1", "N#Cc1cccnc1OC1CCC1", "C#C.CNc1nc2ccccc2o1", "N#Cc1ncccc1OC1CCC1", "OCC=Cc1cn2ccccc2n1", "O=CCCc1cc2ccncc2[nH]1", "Cc1cnc(C...
[ 0.18540075421333313, 0.18008114397525787, 0.17796678841114044, 0.17754021286964417, 0.17681884765625, 0.1765572726726532, 0.17643038928508759, 0.17509472370147705, 0.17439588904380798, 0.17346593737602234, 0.1730617880821228, 0.17290809750556946, 0.1725216954946518, 0.17251013219356537, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,702
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
20
null
null
1,159
4,603
0.117068
O=NCCc1cc2ccccc2[nH]1
0.157805
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "O=CCCc1ccc2nc[nH]c2c1", "C#C.CNc1nc2ccccc2o1", "O=CCCc1ccc2cn[nH]c2c1", "N#CC1(C(=O)c2ccc[nH]2)CCC1", "Cc1ccc2ncccc2c1.N=O", "CC(N=O)c1cc2ccccc2[nH]1", "N#Cc1ccn(CC2CC2)c(=O)c1", "O=CCCc1ccc2[nH]ncc2c1", "N#CC1(C(=O)c2cc[nH]c2)CCC1", "O=CCCc1c...
[ 0.15780538320541382, 0.1506265550851822, 0.14946645498275757, 0.149170383810997, 0.14822596311569214, 0.1469438523054123, 0.1466185599565506, 0.14629924297332764, 0.1454012095928192, 0.14393867552280426, 0.14388291537761688, 0.1435607373714447, 0.14294874668121338, 0.1423042118549347, 0....
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,703
test
CNC(=O)c1cc2ccccc2[nH]1
[M-H]-
null
null
173.07204
60
null
null
364
4,603
0.150261
O=NCCc1cc2ccccc2[nH]1
0.185481
[ "O=NCCc1cc2ccccc2[nH]1", "O=CNCc1cc2ccccc2[nH]1", "OCC=Cc1ccn2ccnc2c1", "N#Cc1ccc(C=O)n1CC1CC1", "Cc1cc(C#N)ncc1OC1CC1", "N#Cc1ccc(N)cc1OC1CC1", "N#Cc1cc(N)ccc1OC1CC1", "N#Cc1cccnc1OC1CCC1", "C#C.CNc1nc2ccccc2o1", "N#Cc1ncccc1OC1CCC1", "OCC=Cc1cn2ccccc2n1", "O=CCCc1cc2ccncc2[nH]1", "Cc1cnc(C...
[ 0.18548065423965454, 0.1801733821630478, 0.17839619517326355, 0.1776740998029709, 0.17686031758785248, 0.17665109038352966, 0.17651766538619995, 0.1750922054052353, 0.1748211681842804, 0.17363595962524414, 0.17340800166130066, 0.1728147566318512, 0.1726135015487671, 0.17258340120315552, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,704
test
CNC(=O)c1cc2ccccc2[nH]1
[M+H]+
null
null
175.08659
20
null
null
442
4,603
0.141423
OCC=Cc1ccn2ccnc2c1
0.169814
[ "OCC=Cc1ccn2ccnc2c1", "CON=Cc1cc2ccccc2[nH]1", "CC(=O)N1C=Nc2ccccc2C1", "OCC=Cc1cn2ccccc2n1", "N#CN1CCOc2ccccc2C1", "C#C.CNc1nc2ccccc2o1", "N#CNCC1Cc2ccccc2O1", "O=NCCc1cc2ccccc2[nH]1", "N#CCNc1ccc2c(c1)CCO2", "CN1N=Cc2ccccc2CC1=O", "C1=CCNC(Oc2ccccn2)=C1", "O=Cc1cccnc1N1CC=CC1", "O=CNN=C1Cc...
[ 0.16981364786624908, 0.16328555345535278, 0.16324350237846375, 0.163163423538208, 0.16245102882385254, 0.16229277849197388, 0.161934033036232, 0.1618404984474182, 0.16177013516426086, 0.16143818199634552, 0.16133317351341248, 0.16095852851867676, 0.16072773933410645, 0.1604417860507965, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,705
test
CNC(=O)c1cc2ccccc2[nH]1
[M+H]+
null
null
175.08659
20
null
null
836
4,603
0.129251
N#CN1CCOc2ccccc2C1
0.1624
[ "N#CN1CCOc2ccccc2C1", "OCC=Cc1ccn2ccnc2c1", "N#CNCC1Cc2ccccc2O1", "C1=CNC(Oc2ccccn2)C=C1", "OCC=Cc1cn2ccccc2n1", "N#CCNc1ccc2c(c1)CCO2", "N#Cc1ccn(CC2CC2)c(=O)c1", "C#C.CNc1nc2ccccc2o1", "N#CN1CCc2c(O)cccc2C1", "CNc1ccc(C2CO2)cc1C#N", "N#Cc1ccccc1OC1CNC1", "O=NCCc1cc2ccccc2[nH]1", "N#Cc1ccc(...
[ 0.1624000072479248, 0.16202709078788757, 0.16053175926208496, 0.15836101770401, 0.15819139778614044, 0.157923623919487, 0.1579229086637497, 0.15777570009231567, 0.15776734054088593, 0.15754465758800507, 0.15582096576690674, 0.1553257256746292, 0.15530599653720856, 0.15498501062393188, 0....
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,706
test
CNC(=O)c1cc2ccccc2[nH]1
[M+H]+
null
null
175.08659
60
null
null
573
4,603
0.142517
O=NCCc1cc2ccccc2[nH]1
0.168821
[ "O=NCCc1cc2ccccc2[nH]1", "C#C.CNc1nc2ccccc2o1", "N#Cc1ccc(N)cc1OC1CC1", "N#Cc1ccn(CC2CC2)c(=O)c1", "N#Cc1cc(N)ccc1OC1CC1", "Cc1cc(C#N)ncc1OC1CC1", "N#Cc1ccc(C=O)n1CC1CC1", "Cc1cnc(C#N)cc1OC1CC1", "CC(N=O)c1cc2ccccc2[nH]1", "OCC=Cc1ccn2ccnc2c1", "N#Cc1cccc(OC2CCC2)n1", "CN(O)c1cnc2ccccc2c1", ...
[ 0.16882102191448212, 0.1673644781112671, 0.16676539182662964, 0.16545383632183075, 0.16527318954467773, 0.16519594192504883, 0.16503095626831055, 0.1645997017621994, 0.1642928272485733, 0.1639638990163803, 0.16377393901348114, 0.16359807550907135, 0.16356401145458221, 0.16350513696670532, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,707
test
CNC(=O)c1cc2ccccc2[nH]1
[M+H]+
null
null
175.08659
15
null
null
1,188
4,603
0.111696
N#CN1CCOc2ccccc2C1
0.163951
[ "N#CN1CCOc2ccccc2C1", "O=NCCc1cc2ccccc2[nH]1", "N#CNCC1Cc2ccccc2O1", "N#Cc1ccccc1OC1CNC1", "OCC=Cc1ccn2ccnc2c1", "OCC=Cc1cn2ccccc2n1", "N#CN1CCc2c(O)cccc2C1", "N#CCN1COc2ccccc2C1", "N#Cc1ccn(CC2CC2)c(=O)c1", "N#Cc1cccn1CC(=O)C1CC1", "N#CN(c1ccccc1)C1COC1", "N#Cc1ccccc1NC1COC1", "N#CCNc1ccc2c...
[ 0.16395129263401031, 0.15889763832092285, 0.15809154510498047, 0.15705619752407074, 0.15659934282302856, 0.1561785340309143, 0.1554570198059082, 0.15419486165046692, 0.15403826534748077, 0.15312924981117249, 0.15251272916793823, 0.1515139937400818, 0.15139183402061462, 0.15115420520305634,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,708
test
CNC(=O)c1cc2ccccc2[nH]1
[M+H]+
null
null
175.08659
20
null
null
1,382
4,603
0.113583
N#CN1CCOc2ccccc2C1
0.168416
[ "N#CN1CCOc2ccccc2C1", "N#Cc1ccccc1OC1CNC1", "O=NCCc1cc2ccccc2[nH]1", "N#CN1CCc2c(O)cccc2C1", "N#CNCC1Cc2ccccc2O1", "OCC=Cc1cn2ccccc2n1", "N#Cc1ccn(CC2CC2)c(=O)c1", "OCC=Cc1ccn2ccnc2c1", "N#CN(c1ccccc1)C1COC1", "N#Cc1ccccc1NC1COC1", "N#CCN1COc2ccccc2C1", "OCC#Cc1ccc(C2CC2)nn1", "N#Cc1cc(N)ccc...
[ 0.16841599345207214, 0.16499044001102448, 0.16292497515678406, 0.16161473095417023, 0.16152139008045197, 0.16105516254901886, 0.16067741811275482, 0.16040536761283875, 0.16034412384033203, 0.15996548533439636, 0.1592732071876526, 0.15919995307922363, 0.15877173840999603, 0.1579149663448333...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,709
test
Cc1nnc(SCC#CCSc2nnc(C)s2)s1
[M+H]+
null
null
314.98611
20
null
null
3
9
0.081429
CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C
0.102144
[ "CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C", "C1=CNC(=C1)N(C(=S)S)N(C2=CC=CN2)C(=S)S", "Cc1nnc(SCC#CCSc2nnc(C)s2)s1", "CC1=CC=NN1C(=S)SSC(=S)N2C(=CC=N2)C", "C1=CN=C(N=C1)SSCCSSC2=NC=CC=N2", "CC1=NN(C=C1)C(=S)SSC(=S)N2C=CC(=N2)C", "CC1=CN(N=C1)C(=S)SSC(=S)N2C=C(C=N2)C", "CSC1=NC2=C(S1)CC3=C(N=CN2)N=C(S3)SC"...
[ 0.10214446485042572, 0.08207490295171738, 0.08142884075641632, 0.07318387925624847, 0.07315612584352493, 0.0647692158818245, 0.06120828911662102, 0.054092634469270706, 0.043633926659822464 ]
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,710
test
Cc1nnc(SCC#CCSc2nnc(C)s2)s1
[M+H]+
null
null
314.98611
20
null
null
2
9
0.081605
CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C
0.102597
[ "CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C", "Cc1nnc(SCC#CCSc2nnc(C)s2)s1", "C1=CNC(=C1)N(C(=S)S)N(C2=CC=CN2)C(=S)S", "C1=CN=C(N=C1)SSCCSSC2=NC=CC=N2", "CC1=CC=NN1C(=S)SSC(=S)N2C(=CC=N2)C", "CC1=NN(C=C1)C(=S)SSC(=S)N2C=CC(=N2)C", "CC1=CN(N=C1)C(=S)SSC(=S)N2C=C(C=N2)C", "CSC1=NC2=C(S1)CC3=C(N=CN2)N=C(S3)SC"...
[ 0.10259702056646347, 0.08160455524921417, 0.08156578242778778, 0.07456232607364655, 0.07241228967905045, 0.06413687765598297, 0.060360901057720184, 0.052924349904060364, 0.04425396770238876 ]
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,711
test
Cc1nnc(SCC#CCSc2nnc(C)s2)s1
[M+H]+
null
null
314.98611
60
null
null
3
9
0.093099
CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C
0.116204
[ "CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C", "C1=CN=C(N=C1)SSCCSSC2=NC=CC=N2", "Cc1nnc(SCC#CCSc2nnc(C)s2)s1", "CC1=CC=NN1C(=S)SSC(=S)N2C(=CC=N2)C", "CC1=NN(C=C1)C(=S)SSC(=S)N2C=CC(=N2)C", "CC1=CN(N=C1)C(=S)SSC(=S)N2C=C(C=N2)C", "C1=CNC(=C1)N(C(=S)S)N(C2=CC=CN2)C(=S)S", "CC1=NN=C(S1)SCC#CCSC2=NN=C(S2)C", ...
[ 0.11620396375656128, 0.11584777384996414, 0.09309906512498856, 0.08311497420072556, 0.07661986351013184, 0.06519180536270142, 0.06428442895412445, 0.059513311833143234, 0.041388437151908875 ]
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,712
test
Cc1nnc(SCC#CCSc2nnc(C)s2)s1
[M+H]+
null
null
314.98611
15
null
null
3
9
0.063727
CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C
0.076835
[ "CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C", "C1=CNC(=C1)N(C(=S)S)N(C2=CC=CN2)C(=S)S", "Cc1nnc(SCC#CCSc2nnc(C)s2)s1", "CC1=CC=NN1C(=S)SSC(=S)N2C(=CC=N2)C", "CC1=CN(N=C1)C(=S)SSC(=S)N2C=C(C=N2)C", "CC1=NN(C=C1)C(=S)SSC(=S)N2C=CC(=N2)C", "C1=CN=C(N=C1)SSCCSSC2=NC=CC=N2", "CSC1=NC2=C(S1)CC3=C(N=CN2)N=C(S3)SC"...
[ 0.07683473080396652, 0.07321300357580185, 0.06372740864753723, 0.05127184838056564, 0.04322562366724014, 0.04039161279797554, 0.03921465203166008, 0.036873020231723785, 0.02603892795741558 ]
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,713
test
Cc1nnc(SCC#CCSc2nnc(C)s2)s1
[M+H]+
null
null
314.98611
20
null
null
3
9
0.067372
CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C
0.081578
[ "CC1=NC(=CC(=S)N1)SSC2=CC(=S)NC(=N2)C", "C1=CNC(=C1)N(C(=S)S)N(C2=CC=CN2)C(=S)S", "Cc1nnc(SCC#CCSc2nnc(C)s2)s1", "CC1=CC=NN1C(=S)SSC(=S)N2C(=CC=N2)C", "CC1=CN(N=C1)C(=S)SSC(=S)N2C=C(C=N2)C", "C1=CN=C(N=C1)SSCCSSC2=NC=CC=N2", "CC1=NN(C=C1)C(=S)SSC(=S)N2C=CC(=N2)C", "CSC1=NC2=C(S1)CC3=C(N=CN2)N=C(S3)SC"...
[ 0.08157826960086823, 0.07510402798652649, 0.06737236678600311, 0.05483011156320572, 0.046370163559913635, 0.04483397677540779, 0.04424673318862915, 0.03974952921271324, 0.029281355440616608 ]
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,714
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
20
null
null
52
964
0.066915
C1=C(C(=O)C(N=C1)CCCBr)N2C=NC=N2
0.089031
[ "C1=C(C(=O)C(N=C1)CCCBr)N2C=NC=N2", "C1=CN2C(=C(C=N2)C(=O)NCCCBr)C=N1", "CNCCC1=NC(=NO1)C2=C(C=CC=N2)Br", "CC(C)NC(=O)C1=C2C=C(C=NC2=NN1)Br", "C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N", "CC1=C(C(=NN1)N2CC(CC2=O)CBr)C#N", "CCCNC(=O)C1=NN2C=C(C=NC2=C1)Br", "CC1=C(N2C=C(C(=C(C2=N1)Br)N)C(=O)N)C", "C1C(C(=NN)NNC1...
[ 0.08903083205223083, 0.0886719673871994, 0.08166657388210297, 0.08028530329465866, 0.08006623387336731, 0.07987417280673981, 0.07947531342506409, 0.0785740315914154, 0.07801677286624908, 0.07768744975328445, 0.0769842192530632, 0.0766804963350296, 0.07622355222702026, 0.07587362825870514, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,715
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
20
null
null
55
964
0.058928
C1=CN2C(=C(C=N2)C(=O)NCCCBr)C=N1
0.077232
[ "C1=CN2C(=C(C=N2)C(=O)NCCCBr)C=N1", "C1=C(C(=O)C(N=C1)CCCBr)N2C=NC=N2", "C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N", "CC(C)NC(=O)C1=C2C=C(C=NC2=NN1)Br", "CNCCC1=NC(=NO1)C2=C(C=CC=N2)Br", "CC1=C(N2C=C(C(=C(C2=N1)Br)N)C(=O)N)C", "CC1=C(N(N=C1C)C2=C(C(=O)NC=N2)Br)C", "CCCNC(=O)C1=NN2C=C(C=NC2=C1)Br", "CCNC(=O)C1=...
[ 0.07723192125558853, 0.07695519179105759, 0.0745934396982193, 0.07379606366157532, 0.07331482321023941, 0.07244269549846649, 0.0717482939362526, 0.07103700935840607, 0.07074236869812012, 0.06991513073444366, 0.06945179402828217, 0.06930401921272278, 0.06926180422306061, 0.06896951794624329...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,716
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
60
null
null
53
964
0.079082
C1=C(C(=O)C(N=C1)CCCBr)N2C=NC=N2
0.113748
[ "C1=C(C(=O)C(N=C1)CCCBr)N2C=NC=N2", "C1=CN2C(=C(C=N2)C(=O)NCCCBr)C=N1", "CC1=C(C(=NN1)N2CC(CC2=O)CBr)C#N", "CN(CCBr)C(=O)C1=C2C=NC=CN2N=C1", "CNCCC1=NC(=NO1)C2=C(C=CC=N2)Br", "CCCNC(=O)C1=NN2C=C(C=NC2=C1)Br", "C1=C(C=NC=C1Br)CNCCC2=NC=NO2", "CN1C=CC(=N1)NN2C=C(C=CC2=O)CBr", "C1C(C(=NN)NNC1=O)C2=CC=C...
[ 0.11374783515930176, 0.11080007255077362, 0.10168828815221786, 0.09802301228046417, 0.09645864367485046, 0.09548228979110718, 0.0945344790816307, 0.09261796623468399, 0.09115899354219437, 0.09094884991645813, 0.09005468338727951, 0.08978895843029022, 0.08927026391029358, 0.0889816284179687...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,717
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
30
null
null
97
964
0.038412
C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N
0.073355
[ "C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N", "CN(C)C1=C(C=C(C=N1)Br)C(=O)NCC#N", "C1=CC(=C(C=C1Br)C#N)NCCNC(=O)N", "C1=CC(=C(C=C1Br)NCCNC(=O)N)C#N", "C1=CC(=C(C=C1C#N)Br)NCCNC(=O)N", "C1=CC(=C(C=C1C#N)Br)NCC(C(=O)N)N", "CCC(C(=O)N)NC1=CC(=C(N=C1)C#N)Br", "C1=CC(=C(C=C1Br)C#N)NCC(C(=O)N)N", "CC1=C(C=C(C=C1)C(=O...
[ 0.07335461676120758, 0.06586271524429321, 0.06481148302555084, 0.06460769474506378, 0.06389785557985306, 0.06245806813240051, 0.061775486916303635, 0.06118437647819519, 0.06062467396259308, 0.059754155576229095, 0.05847081169486046, 0.05796638876199722, 0.05795922875404358, 0.0574212409555...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,718
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
20
null
null
71
964
0.043589
CC1=C(N(N=C1C)C2=C(C(=O)NC=N2)Br)C
0.062196
[ "CC1=C(N(N=C1C)C2=C(C(=O)NC=N2)Br)C", "CC1=C(N2C=C(C(=C(C2=N1)Br)N)C(=O)N)C", "CC(C)NC(=O)C1=C2C=C(C=NC2=NN1)Br", "C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N", "CC(C)C1=NC(=C2N1C(=CN=C2N)C=O)Br", "CCNC(=O)C1=C(N2C=CC=C(C2=N1)Br)N", "CC1=NC=C(C(=O)N1CCN2C=CC=N2)Br", "CNCCC1=NC(=NO1)C2=C(C=CC=N2)Br", "CCN1C(=O)C(...
[ 0.062195755541324615, 0.06151241809129715, 0.060070183128118515, 0.05963902547955513, 0.05856361985206604, 0.05722885578870773, 0.05693181976675987, 0.055989522486925125, 0.0553458072245121, 0.05504738166928291, 0.05493089556694031, 0.054825037717819214, 0.05374350771307945, 0.053726539015...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,719
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
60
null
null
53
964
0.079083
C1=C(C(=O)C(N=C1)CCCBr)N2C=NC=N2
0.113748
[ "C1=C(C(=O)C(N=C1)CCCBr)N2C=NC=N2", "C1=CN2C(=C(C=N2)C(=O)NCCCBr)C=N1", "CC1=C(C(=NN1)N2CC(CC2=O)CBr)C#N", "CN(CCBr)C(=O)C1=C2C=NC=CN2N=C1", "CNCCC1=NC(=NO1)C2=C(C=CC=N2)Br", "CCCNC(=O)C1=NN2C=C(C=NC2=C1)Br", "C1=C(C=NC=C1Br)CNCCC2=NC=NO2", "CN1C=CC(=N1)NN2C=C(C=CC2=O)CBr", "C1C(C(=NN)NNC1=O)C2=CC=C...
[ 0.1137482076883316, 0.1108003631234169, 0.10168872773647308, 0.09802325814962387, 0.09645970165729523, 0.09548303484916687, 0.09453524649143219, 0.09261885285377502, 0.09115948528051376, 0.09094975888729095, 0.09005531668663025, 0.08978965878486633, 0.08927066624164581, 0.08898245543241501...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,720
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
30
null
null
97
964
0.03841
C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N
0.07271
[ "C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N", "CN(C)C1=C(C=C(C=N1)Br)C(=O)NCC#N", "C1=CC(=C(C=C1Br)C#N)NCCNC(=O)N", "C1=CC(=C(C=C1Br)NCCNC(=O)N)C#N", "C1=CC(=C(C=C1C#N)Br)NCCNC(=O)N", "C1=CC(=C(C=C1C#N)Br)NCC(C(=O)N)N", "CCC(C(=O)N)NC1=CC(=C(N=C1)C#N)Br", "C1=CC(=C(C=C1Br)C#N)NCC(C(=O)N)N", "CC1=C(C=C(C=C1)C(=O...
[ 0.07271003723144531, 0.06531738489866257, 0.06418121606111526, 0.0639757513999939, 0.06325722485780716, 0.06188516318798065, 0.061193373054265976, 0.0606226809322834, 0.06002335250377655, 0.059075988829135895, 0.05826294794678688, 0.057953719049692154, 0.057346493005752563, 0.0573172420263...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,721
test
COCCn1cc(-c2cc(Br)cnc2)nn1
[M+H]+
null
null
283.0189
20
null
null
71
964
0.043595
CC1=C(N(N=C1C)C2=C(C(=O)NC=N2)Br)C
0.062205
[ "CC1=C(N(N=C1C)C2=C(C(=O)NC=N2)Br)C", "CC1=C(N2C=C(C(=C(C2=N1)Br)N)C(=O)N)C", "CC(C)NC(=O)C1=C2C=C(C=NC2=NN1)Br", "C1=CC(=C(C=C1NCCNC(=O)N)Br)C#N", "CC(C)C1=NC(=C2N1C(=CN=C2N)C=O)Br", "CCNC(=O)C1=C(N2C=CC=C(C2=N1)Br)N", "CC1=NC=C(C(=O)N1CCN2C=CC=N2)Br", "CNCCC1=NC(=NO1)C2=C(C=CC=N2)Br", "CCN1C(=O)C(...
[ 0.06220458447933197, 0.061520420014858246, 0.06007373332977295, 0.059613972902297974, 0.05857796221971512, 0.05723387748003006, 0.05693615600466728, 0.05598627030849457, 0.05534527450799942, 0.055059440433979034, 0.0549122616648674, 0.054831843823194504, 0.05373966321349144, 0.053730729967...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,722
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+Cl]-
null
null
305.02137
20
null
null
116
298
0.084792
CC1=NN(C(=C1CN2C(=O)C(=O)N(C2=O)C)Cl)C
0.132161
[ "CC1=NN(C(=C1CN2C(=O)C(=O)N(C2=O)C)Cl)C", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "C1CCN(C1)C(=O)NC(=O)C2=CC(=NNC2=O)Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CC1C(=O)NC(=O)CN1C2=C(C(=NC=N2)Cl)OC", "CC(C)C1=NC(=NO1)CN2C=C(C(=O)NC2=O)Cl", "CN1C(=CN=C1CN2C(=O)...
[ 0.1321614682674408, 0.13088345527648926, 0.13042861223220825, 0.129582941532135, 0.12779316306114197, 0.1178211197257042, 0.11652053147554398, 0.11570168286561966, 0.11537973582744598, 0.11511295288801193, 0.11498714983463287, 0.11489318311214447, 0.11455672979354858, 0.11447714269161224, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,723
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+Cl]-
null
null
305.02137
20
null
null
105
298
0.070323
CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C
0.114406
[ "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CC1=NN(C(=C1CN2C(=O)C(=O)N(C2=O)C)Cl)C", "C1CCN(C1)C(=O)NC(=O)C2=CC(=NNC2=O)Cl", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC(C)(C)OC(=O)N1C(=...
[ 0.11440597474575043, 0.11413263529539108, 0.11384208500385284, 0.11307165026664734, 0.1089782565832138, 0.10387293994426727, 0.10234258323907852, 0.10228550434112549, 0.09922351688146591, 0.0988011509180069, 0.09804695844650269, 0.09790749847888947, 0.09731785953044891, 0.09665931761264801...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,724
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+Cl]-
null
null
305.02137
60
null
null
104
298
0.075672
CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl
0.12021
[ "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "CC1=NN(C(=C1CN2C(=O)C(=O)N(C2=O)C)Cl)C", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "C1CCN(C1)C(=O)NC(=O)C2=CC(=NNC2=O)Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC1C(=O)NC(=O)CN1C2...
[ 0.12020984292030334, 0.11967755109071732, 0.11869914084672928, 0.11840067058801651, 0.11736010015010834, 0.10675463825464249, 0.10629472136497498, 0.10525336861610413, 0.10426817834377289, 0.10379710793495178, 0.10307327657938004, 0.10280340164899826, 0.10271142423152924, 0.101485982537269...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,725
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+Cl]-
null
null
305.02137
15
null
null
104
298
0.06958
CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C
0.113578
[ "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CC1=NN(C(=C1CN2C(=O)C(=O)N(C2=O)C)Cl)C", "C1CCN(C1)C(=O)NC(=O)C2=CC(=NNC2=O)Cl", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC(C)(C)OC(=O)N1C(=...
[ 0.11357846856117249, 0.11330883204936981, 0.11255009472370148, 0.11183779686689377, 0.10816644132137299, 0.10311846435070038, 0.10164061188697815, 0.10143949091434479, 0.0984189510345459, 0.09784519672393799, 0.09720789641141891, 0.09678395092487335, 0.09631245583295822, 0.0957256704568862...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,726
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+Cl]-
null
null
305.02137
20
null
null
103
298
0.073777
CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl
0.11788
[ "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CC1=NN(C(=C1CN2C(=O)C(=O)N(C2=O)C)Cl)C", "C1CCN(C1)C(=O)NC(=O)C2=CC(=NNC2=O)Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC1C(=O)NC(=O)CN1C2...
[ 0.11787975579500198, 0.11690245568752289, 0.11636856198310852, 0.11528877913951874, 0.11447449773550034, 0.10539371520280838, 0.10488561540842056, 0.10254277288913727, 0.10199525207281113, 0.1008158028125763, 0.10059931874275208, 0.10032563656568527, 0.10000587999820709, 0.0994382128119468...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,727
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+FA]-
null
null
315.05017
20
null
null
120
298
0.06703
COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl
0.11597
[ "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "CC1=NN(C(=C1CN2C(=O)C(=O)N(C2=O)C)Cl)C", "CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "C1CCN(C1)C(=O)NC(=O)C2=CC(=NNC2=O)Cl", "CCC1C(=O)NC(=O)CN...
[ 0.11597011983394623, 0.11312147229909897, 0.11255103349685669, 0.11018826067447662, 0.10410493612289429, 0.1038876473903656, 0.10336257517337799, 0.10110890865325928, 0.10051359981298447, 0.09806704521179199, 0.09737280011177063, 0.09686070680618286, 0.09645041078329086, 0.0963184833526611...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,728
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+FA]-
null
null
315.05017
20
null
null
96
298
0.03977
CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl
0.086445
[ "CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl", "CC(=O)CN1C2=C(C(=O)N(C(=O)N2C)C)N=C1Cl", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC1=NN(C(=C1CN2C(...
[ 0.08644506335258484, 0.08072738349437714, 0.08054011315107346, 0.08021461963653564, 0.07577547430992126, 0.07503679394721985, 0.07151482999324799, 0.07045421749353409, 0.06919404119253159, 0.06716721504926682, 0.06650791317224503, 0.06416049599647522, 0.06326507031917572, 0.061381004750728...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,729
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+FA]-
null
null
315.05017
60
null
null
99
298
0.029605
CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl
0.07985
[ "CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl", "CC(=O)CN1C2=C(C(=O)N(C(=O)N2C)C)N=C1Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC(C(=O)Cl)N1C=NC...
[ 0.07985042035579681, 0.07422114163637161, 0.06912537664175034, 0.068252794444561, 0.0656164363026619, 0.061471618711948395, 0.060412466526031494, 0.05946830287575722, 0.057848185300827026, 0.05573378875851631, 0.05505264177918434, 0.05248461663722992, 0.05226628854870796, 0.052242904901504...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,730
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+FA]-
null
null
315.05017
15
null
null
96
298
0.039098
CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl
0.087
[ "CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl", "CC(=O)CN1C2=C(C(=O)N(C(=O)N2C)C)N=C1Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC1=NN(C(=C1CN2C(...
[ 0.08700025826692581, 0.08147270232439041, 0.08010853826999664, 0.07952626049518585, 0.0752425491809845, 0.07370127737522125, 0.07072117179632187, 0.06913035362958908, 0.06890405714511871, 0.06674765795469284, 0.06566518545150757, 0.0632840096950531, 0.0626705214381218, 0.06129726767539978,...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,731
test
OCC1OC(n2cnc3c(Cl)ncnc32)CC1O
[M+FA]-
null
null
315.05017
20
null
null
101
298
0.035387
CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl
0.084325
[ "CC(C)(C)OC(=O)N1C(=O)N2C=CN=C(C2=N1)Cl", "CC(=O)CN1C2=C(C(=O)N(C(=O)N2C)C)N=C1Cl", "COCCN1C=C(C=N1)N2C(=O)C=C(NC2=O)Cl", "CC1(C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl)C", "CN1C(=O)CCC(C1=O)NC2=C(C(=O)NC=N2)Cl", "CN1C(=O)C(=C(C=N1)NC2CCC(=O)NC2=O)Cl", "CCC1C(=O)NC(=O)CN1C2=C(C(=O)NC=N2)Cl", "CC(C(=O)Cl)N1C=NC...
[ 0.08432495594024658, 0.07890278100967407, 0.07707835733890533, 0.07609929889440536, 0.07238104939460754, 0.0702541247010231, 0.06745648384094238, 0.06578952074050903, 0.0645989254117012, 0.06408896297216415, 0.0621570460498333, 0.05960514396429062, 0.05934104323387146, 0.058247581124305725...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,732
test
Cc1c(I)c(C2C=CNC=N2)c(C)s1
[M+H]+
null
null
318.97604
20
null
null
5
71
0.061274
C1=CC=C2C(=C1)N=C(S2)NCCCI
0.086716
[ "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "C1C(=NCCI)NC2=CC=CC=C2S1", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "Cc1c(I)c(C2C=CNC=N2)c(C)s1", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "C[N+]1=CN=C(C2=CC=CC=C21)SC.[I-]", "C1=CC=C2C(=C1)N=C(S2)CNCCI", "CC1=CSC(=N1)C2=C[N+](=CC=C2)C.[I-]", "CC1=NC(...
[ 0.08671589940786362, 0.07982626557350159, 0.0741972029209137, 0.06138104572892189, 0.06127424165606499, 0.061226800084114075, 0.05982659384608269, 0.05943369120359421, 0.05780516564846039, 0.05702269822359085, 0.05601547285914421, 0.05451909825205803, 0.05060916393995285, 0.049879483878612...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,733
test
Cc1c(I)c(C2C=CNC=N2)c(C)s1
[M+H]+
null
null
318.97604
20
null
null
6
71
0.055398
C1=CC=C2C(=C1)N=C(S2)NCCCI
0.081041
[ "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "C1C(=NCCI)NC2=CC=CC=C2S1", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "Cc1c(I)c(C2C=CNC=N2)c(C)s1", "C[N+]1=CN=C(C2=CC=CC=C21)SC.[I-]", "C1=CC=C2C(=C1)N=C(S2)CNCCI", "CC1=CSC(=N1)C2=C[N+](=CC=C2)C.[I-]", "CC1=NC(...
[ 0.08104070276021957, 0.07428926229476929, 0.070004902780056, 0.056421175599098206, 0.05566089227795601, 0.055397965013980865, 0.053887370973825455, 0.05206969007849693, 0.050888918340206146, 0.05045172572135925, 0.04926953464746475, 0.046966634690761566, 0.045056652277708054, 0.04442167282...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,734
test
Cc1c(I)c(C2C=CNC=N2)c(C)s1
[M+H]+
null
null
318.97604
60
null
null
19
71
0.033787
C1C(=NCCI)NC2=CC=CC=C2S1
0.104321
[ "C1C(=NCCI)NC2=CC=CC=C2S1", "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "CC1=CC(=C2C(=C1N)C=CN2SI)C", "C1CN(C2=CC=CC=C2C=C1N)SI", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "CC1=NC(=CS1)C2=C[N+](=CC=C2)C.[I-]", "CC1=CSC(=N1)C2=C[N+](=CC=C2)C.[I-]", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "CN(C)C1...
[ 0.10432089865207672, 0.08944512158632278, 0.08298084884881973, 0.0786500796675682, 0.07506321370601654, 0.07042565941810608, 0.0665787011384964, 0.06553616374731064, 0.06110042706131935, 0.05987244471907616, 0.05655823275446892, 0.053889550268650055, 0.0535854734480381, 0.05297031253576279...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,735
test
Cc1c(I)c(C2C=CNC=N2)c(C)s1
[M+H]+
null
null
318.97604
20
null
null
3
71
0.065279
CC(C)N1C2=C(C=C(C=C2)I)NC1=S
0.075474
[ "CC(C)N1C2=C(C=C(C=C2)I)NC1=S", "C1=CC=C2C(=C1)N=C(S2)NCCCI", "Cc1c(I)c(C2C=CNC=N2)c(C)s1", "CC(C)(C)C1=C2C=CSC2=NC(=N1)I", "CC(C)N1C=C(C(=N1)C2=CC=CS2)I", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "CC(C)N1C(=C(C=N1)I)C2=CC=CS2", "CC(C)N1C=C(C(=N1)C2=CSC=C2)I", "CC1=C(C(=C(S1)C)I)C2C=CNC=N2", "CC(C)C1=C(C=C...
[ 0.075474314391613, 0.06662171334028244, 0.06527919322252274, 0.061630286276340485, 0.06088992953300476, 0.059028152376413345, 0.05547437071800232, 0.0541815459728241, 0.052403490990400314, 0.05124349519610405, 0.04971279203891754, 0.04724044352769852, 0.047165073454380035, 0.04699998348951...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,736
test
Cc1c(I)c(C2C=CNC=N2)c(C)s1
[M+H]+
null
null
318.97604
45
null
null
18
71
0.029783
C1C(=NCCI)NC2=CC=CC=C2S1
0.094404
[ "C1C(=NCCI)NC2=CC=CC=C2S1", "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "CC1=CC(=C2C(=C1N)C=CN2SI)C", "C1CN(C2=CC=CC=C2C=C1N)SI", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "CC1=NC(=CS1)C2=C[N+](=CC=C2)C.[I-]", "CC1=CSC(=N1)C2=C[N+](=CC=C2)C.[I-]", "C[N+]1=...
[ 0.09440404921770096, 0.08286137878894806, 0.07320123165845871, 0.06254901736974716, 0.06247120723128319, 0.05664832890033722, 0.05279674008488655, 0.05270043760538101, 0.051328420639038086, 0.04555683583021164, 0.04314928501844406, 0.042614761739969254, 0.04099886864423752, 0.0403041951358...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,737
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
20
null
null
27
71
0.035335
C1=CC=C2C(=C1)N=C(S2)NCCCI
0.085442
[ "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "C1C(=NCCI)NC2=CC=CC=C2S1", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "C1=CC=C2C(=C1)N=C(S2)CNCCI", "CC(C)N1C2=C(C=C(C=C2)I)NC1=S", "C[N+]1=CN=C(C2=CC=CC=C21)SC.[I-]", "CC(C)N1C=C(C(=N1)C2=CC=CS2)I", "CC(C)N1C(=C...
[ 0.08544186502695084, 0.07699059695005417, 0.07219358533620834, 0.05989696830511093, 0.05762780085206032, 0.057248905301094055, 0.05660218000411987, 0.0558767206966877, 0.05172150582075119, 0.05087781324982643, 0.05054885894060135, 0.05040818825364113, 0.05001536384224892, 0.049241468310356...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,738
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
20
null
null
26
71
0.027694
C1=CC=C2C(=C1)N=C(S2)NCCCI
0.077213
[ "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "C1C(=NCCI)NC2=CC=CC=C2S1", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "CC(C)N1C2=C(C=C(C=C2)I)NC1=S", "C[N+]1=CN=C(C2=CC=CC=C21)SC.[I-]", "C1=CC=C2C(=C1)N=C(S2)CNCCI", "CC(C)N1C(=C(C=N1)I)C2=CC=CS2", "CC(C)N1C=C(...
[ 0.07721253484487534, 0.06861065328121185, 0.06519687175750732, 0.052577905356884, 0.04917101562023163, 0.047820914536714554, 0.04731421917676926, 0.046968087553977966, 0.04459688067436218, 0.044131528586149216, 0.041778337210416794, 0.04000651463866234, 0.03996497392654419, 0.0398320183157...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,739
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
60
null
null
59
71
-0.013822
C1C(=NCCI)NC2=CC=CC=C2S1
0.099811
[ "C1C(=NCCI)NC2=CC=CC=C2S1", "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "CC1=CC(=C2C(=C1N)C=CN2SI)C", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "C1CN(C2=CC=CC=C2C=C1N)SI", "CC1=NC(=CS1)C2=C[N+](=CC=C2)C.[I-]", "CC1=CSC(=N1)C2=C[N+](=CC=C2)C.[I-]", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "CN(C)C1...
[ 0.09981130063533783, 0.08622832596302032, 0.07863327860832214, 0.07137463986873627, 0.06649556756019592, 0.06639635562896729, 0.058412328362464905, 0.05718138813972473, 0.05572700873017311, 0.05023479461669922, 0.048342447727918625, 0.04754548519849777, 0.04733487591147423, 0.0463804341852...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,740
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
30
null
null
29
71
0.026422
C1=CC=C2C(=C1)N=C(S2)NCCCI
0.07861
[ "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "C1C(=NCCI)NC2=CC=CC=C2S1", "CC(C)N1C2=C(C=C(C=C2)I)NC1=S", "C1=CC=C2C(=C1)N=C(S2)CNCCI", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "C[N+]1=CN=C(C2=CC=CC=C21)SC.[I-]", "CC(C)N1C=C(C(=N1)C2=CC=CS2)I", "CC1=CSC(=N1...
[ 0.0786096602678299, 0.06938496232032776, 0.063088059425354, 0.051713235676288605, 0.05090215802192688, 0.050387196242809296, 0.05011526495218277, 0.04935232177376747, 0.04493970423936844, 0.04310526326298714, 0.04237618297338486, 0.04213515669107437, 0.04066799581050873, 0.0396652445197105...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,741
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
20
null
null
5
71
0.056638
CC(C)N1C2=C(C=C(C=C2)I)NC1=S
0.079408
[ "CC(C)N1C2=C(C=C(C=C2)I)NC1=S", "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC(C)(C)C1=C2C=CSC2=NC(=N1)I", "CC(C)N1C=C(C(=N1)C2=CC=CS2)I", "Cc1sc(C)c(C2C=CNC=N2)c1I", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "CC(C)N1C=C(C(=N1)C2=CSC=C2)I", "CC(C)C1=C(C=CC2=C1N=C(S2)N)I", "CC(C)N1C(=C(C=N1)I)C2=CC=CS2", "C1=CC2=C(C=C1I)...
[ 0.07940837740898132, 0.06289436668157578, 0.06198783591389656, 0.061196912080049515, 0.05663815885782242, 0.055636823177337646, 0.055483754724264145, 0.054371245205402374, 0.05167558044195175, 0.05092840641736984, 0.050686322152614594, 0.05038106068968773, 0.045884933322668076, 0.044921230...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,742
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
60
null
null
59
71
-0.013709
C1C(=NCCI)NC2=CC=CC=C2S1
0.100146
[ "C1C(=NCCI)NC2=CC=CC=C2S1", "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "CC1=CC(=C2C(=C1N)C=CN2SI)C", "C1CN(C2=CC=CC=C2C=C1N)SI", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "CC1=NC(=CS1)C2=C[N+](=CC=C2)C.[I-]", "CC1=CSC(=N1)C2=C[N+](=CC=C2)C.[I-]", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "CN(C)C1...
[ 0.10014638304710388, 0.0864839106798172, 0.07897745817899704, 0.07192417979240417, 0.06711553037166595, 0.06674478948116302, 0.059091731905937195, 0.05789899453520775, 0.05613406002521515, 0.05096198245882988, 0.04877906292676926, 0.0478053018450737, 0.04777347669005394, 0.0470778979361057...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,743
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
30
null
null
29
71
0.026571
C1=CC=C2C(=C1)N=C(S2)NCCCI
0.078786
[ "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "C1C(=NCCI)NC2=CC=CC=C2S1", "CC(C)N1C2=C(C=C(C=C2)I)NC1=S", "C1=CC=C2C(=C1)N=C(S2)CNCCI", "C1C(SC(=N1)NC2=CC=CC=C2)CI", "C[N+]1=NC=C(C2=CC=CC=C21)SC.[I-]", "C[N+]1=CN=C(C2=CC=CC=C21)SC.[I-]", "CC(C)N1C=C(C(=N1)C2=CC=CS2)I", "CC1=CSC(=N1...
[ 0.07878568768501282, 0.06958243250846863, 0.06326784938573837, 0.05189008638262749, 0.05114862322807312, 0.05053061246871948, 0.05034859478473663, 0.04960508644580841, 0.04506765305995941, 0.043468963354825974, 0.042649585753679276, 0.042476195842027664, 0.040755510330200195, 0.03979770839...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,744
test
Cc1sc(C)c(C2C=CNC=N2)c1I
[M+H]+
null
null
318.97604
20
null
null
5
71
0.056727
CC(C)N1C2=C(C=C(C=C2)I)NC1=S
0.079599
[ "CC(C)N1C2=C(C=C(C=C2)I)NC1=S", "C1=CC=C2C(=C1)N=C(S2)NCCCI", "CC(C)(C)C1=C2C=CSC2=NC(=N1)I", "CC(C)N1C=C(C(=N1)C2=CC=CS2)I", "Cc1sc(C)c(C2C=CNC=N2)c1I", "CC1=CC(=C(C2=C1N=C(S2)N)C)CI", "CC(C)N1C=C(C(=N1)C2=CSC=C2)I", "CC(C)C1=C(C=CC2=C1N=C(S2)N)I", "CC(C)N1C(=C(C=N1)I)C2=CC=CS2", "C1=CC2=C(C=C1I)...
[ 0.07959876954555511, 0.06311528384685516, 0.062196847051382065, 0.06138617545366287, 0.05672673135995865, 0.055834267288446426, 0.05567809194326401, 0.054541438817977905, 0.05186370015144348, 0.0512043759226799, 0.050870537757873535, 0.0505903922021389, 0.046162206679582596, 0.045067314058...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,745
test
COC(=O)c1sccc1NC(=O)CSc1nnnn1C
[M+H]+
null
null
314.03761
20
null
null
1
148
0.119503
COC(=O)c1sccc1NC(=O)CSc1nnnn1C
0.119503
[ "COC(=O)c1sccc1NC(=O)CSc1nnnn1C", "CN1C(=NC(=O)C(=O)N1)SCC2=C(SC=C2)C(=O)NN", "CN1C(=NC(=O)C(=O)N1)SCC2=CC=C(S2)C(=O)NN", "C1=CN(C(=S)NC1=O)CNOCC2=CNC(=S)NC2=O", "C1=CSC(=C1)CN2C(=NN=N2)SCC(=O)NCC(=O)O", "CC1C(=O)N=C(S1)NC(=O)CSC2=NC(=O)CC(=N2)N", "CC1=NN=C(S1)SCC(=O)C2=C(N(C(=O)NC2=O)C)N", "C1=CC(=CC...
[ 0.11950299143791199, 0.11575897783041, 0.09596746414899826, 0.09484948217868805, 0.09386542439460754, 0.09309511631727219, 0.08638117462396622, 0.0852418765425682, 0.08512154221534729, 0.08359567821025848, 0.0828823372721672, 0.08206593990325928, 0.08135490864515305, 0.07880931347608566, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1
502,746
test
COC(=O)c1sccc1NC(=O)CSc1nnnn1C
[M+H]+
null
null
314.03761
20
null
null
1
148
0.106152
COC(=O)c1sccc1NC(=O)CSc1nnnn1C
0.106152
[ "COC(=O)c1sccc1NC(=O)CSc1nnnn1C", "CN1C(=NC(=O)C(=O)N1)SCC2=C(SC=C2)C(=O)NN", "CN1C(=NC(=O)C(=O)N1)SCC2=CC=C(S2)C(=O)NN", "C1=CN(C(=S)NC1=O)CNOCC2=CNC(=S)NC2=O", "CC1C(=O)N=C(S1)NC(=O)CSC2=NC(=O)CC(=N2)N", "C1=CSC(=C1)CN2C(=NN=N2)SCC(=O)NCC(=O)O", "CC1=NN=C(S1)SCC(=O)C2=C(N(C(=O)NC2=O)C)N", "CC1=NN=C(...
[ 0.10615178197622299, 0.10606236755847931, 0.08659794926643372, 0.08515642583370209, 0.0823921486735344, 0.0789722129702568, 0.07722398638725281, 0.0757620707154274, 0.0748804435133934, 0.07200190424919128, 0.0717339813709259, 0.06996864080429077, 0.06844423711299896, 0.0668497160077095, ...
ultrams_codebook
UltraMS codebook
spectrum-encoder-to-ChemBERTa cosine
0
score descending, then frozen candidate position ascending
1