| | |
| | 4llx 1.75 2014 2.89 Ki=1300uM 1 |
| | 5c28 1.56 2015 5.66 Ki=2.2uM 1 |
| | 3uuo 2.11 2012 7.96 Ki=11nM 1 |
| | 3ui7 2.28 2011 9.00 Ki=1nM 1 |
| | 5c2h 2.09 2015 11.09 Ki=8.2pM 1 |
| | 2v00 1.55 2007 3.66 Kd=0.22mM 2 |
| | 3wz8 1.45 2015 5.82 Ki=1.5uM 2 |
| | 3pww 1.22 2011 7.32 Ki=48nM 2 |
| | 3prs 1.38 2011 7.82 Ki=15nM 2 |
| | 3uri 2.10 2012 9.00 Ki=1nM 2 |
| | 4m0z 2.00 2014 5.19 Kd=6.4uM 3 |
| | 4m0y 1.70 2014 6.46 Kd=0.35uM 3 |
| | 3qgy 2.10 2011 7.80 Ki=16nM 3 |
| | 4qd6 2.45 2015 8.64 Ki=2.3nM 3 |
| | 4rfm 2.10 2015 10.05 Ki=90pM 3 |
| | 4cr9 1.70 2015 4.10 Ki=80uM 4 |
| | 4cra 1.80 2015 7.22 Ki=0.06uM 4 |
| | 4x6p 1.93 2015 8.30 Ki=5nM 4 |
| | 4crc 1.60 2015 8.72 Ki=0.0019uM 4 |
| | 4ty7 2.09 2014 9.52 Ki=0.3nM 4 |
| | 5aba 1.62 2015 2.98 Kd=1040uM 5 |
| | 5a7b 1.40 2015 3.57 Kd=271uM 5 |
| | 4agn 1.60 2012 3.97 Kd=107uM 5 |
| | 4agp 1.50 2012 4.69 Kd=20.6uM 5 |
| | 4agq 1.42 2012 5.01 Kd=9.7uM 5 |
| | 3bgz 2.40 2007 6.26 Ki=0.55uM 6 |
| | 3jya 2.10 2009 6.89 Ki=0.1301uM 6 |
| | 2c3i 1.90 2005 7.60 Kd=25nM 6 |
| | 4k18 2.05 2013 8.96 Ki=1.1nM 6 |
| | 5dwr 2.00 2015 11.22 Ki=6pM 6 |
| | 3mss 1.95 2010 4.66 Kd=22uM 7 |
| | 3k5v 1.74 2010 6.30 Kd=0.5uM 7 |
| | 3pyy 1.85 2011 6.86 Kd=137nM 7 |
| | 2v7a 2.50 2007 8.30 Kd=0.005uM 7 |
| | 4twp 2.40 2015 10.00 Ki=100pM 7 |
| | 3wtj 2.24 2015 6.53 Kd=0.297uM 8 |
| | 3zdg 2.48 2013 7.10 Ki=79nM 8 |
| | 3u8k 2.47 2011 8.66 Ki=2.2nM 8 |
| | 4qac 2.10 2014 9.40 Kd=0.4nM 8 |
| | 3u8n 2.35 2011 10.17 Ki=0.067nM 8 |
| | 1a30 2.00 1998 4.30 Ki=50uM 9 |
| | 2qnq 2.30 2008 6.11 Ki=0.77uM 9 |
| | 1g2k 1.95 2001 7.96 Ki=11nM 9 |
| | 1eby 2.29 2002 9.70 Ki=0.20nM 9 |
| | 3o9i 1.45 2011 11.82 Ki=1.5pM 9 |
| | 4lzs 2.20 2014 4.80 Kd=16uM 10 |
| | 3u5j 1.60 2011 5.61 Kd=2.46uM 10 |
| | 4wiv 1.56 2014 6.26 Kd=550nM 10 |
| | 4ogj 1.65 2014 6.79 Kd=164nM 10 |
| | 3p5o 1.60 2010 7.30 Kd=50.5nM 10 |
| | 1ps3 1.80 2003 2.28 Ki=5.2mM 11 |
| | 3dx1 1.21 2009 3.58 Ki=265uM 11 |
| | 3d4z 1.39 2008 4.89 Ki=13uM 11 |
| | 3dx2 1.40 2009 6.82 Ki=150nM 11 |
| | 3ejr 1.27 2009 8.57 Ki=2.7nM 11 |
| | 3l7b 2.00 2010 2.40 Ki=4.01mM 12 |
| | 4eky 2.45 2012 3.52 Ki=303.0uM 12 |
| | 3g2n 2.10 2010 4.09 Ki=81uM 12 |
| | 3syr 2.40 2012 5.10 Ki=7.9uM 12 |
| | 3ebp 2.00 2009 5.91 Ki=1.24uM 12 |
| | 2w66 2.27 2009 4.05 Ki=89uM 13 |
| | 2w4x 2.42 2009 4.85 Kd=14uM 13 |
| | 2wca 2.30 2009 5.60 Ki=2.5uM 13 |
| | 2xj7 2.00 2010 6.66 Ki=220nM 13 |
| | 2vvn 1.85 2008 7.30 Kd=50nM 13 |
| | 3aru 1.90 2011 3.22 Kd=600uM 14 |
| | 3arv 1.50 2011 5.64 Kd=2.3uM 14 |
| | 3ary 1.35 2011 6.00 Kd=1.0uM 14 |
| | 3arq 1.50 2011 6.40 Kd=0.4uM 14 |
| | 3arp 1.55 2011 7.15 Kd=0.07uM 14 |
| | 4ih5 1.90 2013 4.11 Kd=78uM 15 |
| | 4ih7 2.30 2013 5.24 Kd=5.8uM 15 |
| | 3cj4 2.07 2008 6.51 Kd=0.31uM 15 |
| | 4eo8 1.80 2012 8.15 Kd=7nM 15 |
| | 3gnw 2.39 2009 9.10 Kd=0.79nM 15 |
| | 1gpk 2.10 2002 5.37 Ki=4.3uM 16 |
| | 1gpn 2.35 2002 6.48 Ki=0.334uM 16 |
| | 1h23 2.15 2002 8.35 Ki=4.5nM 16 |
| | 1h22 2.15 2002 9.10 Ki=0.8nM 16 |
| | 1e66 2.10 2001 9.89 Ki=0.13nM 16 |
| | 3f3a 2.00 2008 4.19 Ki=64.8uM 17 |
| | 3f3c 2.10 2008 6.02 Ki=950nM 17 |
| | 4mme 2.50 2013 6.50 Kd=318nM 17 |
| | 3f3d 2.30 2008 7.16 Kd=69nM 17 |
| | 3f3e 1.80 2008 7.70 Kd=20nM 17 |
| | 2wbg 1.85 2009 4.45 Ki=35.2uM 18 |
| | 2cbv 1.95 2006 5.48 Kd=3.3uM 18 |
| | 2j78 1.65 2006 6.42 Kd=384nM 18 |
| | 2j7h 1.95 2006 7.19 Kd=65nM 18 |
| | 2cet 1.97 2006 8.02 Kd=9.6nM 18 |
| | 3udh 1.70 2012 2.85 Kd=1.4mM 19 |
| | 3rsx 2.48 2011 4.41 Kd=38.8uM 19 |
| | 4djv 1.73 2012 6.72 Ki=0.19uM 19 |
| | 2vkm 2.05 2008 8.74 Ki=1.8nM 19 |
| | 4gid 2.00 2012 10.77 Ki=0.017nM 19 |
| | 4jfs 2.00 2013 5.27 Ki=5.4uM 20 |
| | 4j28 1.73 2013 5.70 Ki=2.0uM 20 |
| | 2wvt 1.80 2010 6.12 Kd=755nM 20 |
| | 2xii 1.80 2010 7.20 Kd=63.3nM 20 |
| | 4pcs 1.77 2014 7.85 Ki=14nM 20 |
| | 3rr4 1.68 2012 4.55 Ki=28.05uM 21 |
| | 1s38 1.81 2004 5.15 Ki=7.0uM 21 |
| | 1r5y 1.20 2004 6.46 Ki=0.35uM 21 |
| | 3gc5 1.40 2009 7.26 Ki=55nM 21 |
| | 3ge7 1.50 2009 8.70 Ki=2nM 21 |
| | 4dli 1.91 2013 5.62 Kd=2.40uM 22 |
| | 2zb1 2.50 2008 6.32 Kd=0.48uM 22 |
| | 4f9w 2.00 2013 6.94 Ki=114nM 22 |
| | 3e92 2.00 2008 8.00 Ki=10nM 22 |
| | 3e93 2.00 2008 8.85 Ki=1.4nM 22 |
| | 4owm 1.99 2014 2.96 Ki=1090uM 23 |
| | 3twp 1.83 2012 3.92 Ki=119uM 23 |
| | 3r88 1.73 2012 4.82 Ki=15uM 23 |
| | 4gkm 1.67 2013 5.17 Ki=6.8uM 23 |
| | 3qqs 1.97 2012 5.82 Ki=1.5uM 23 |
| | 3gv9 1.80 2009 2.12 Ki=7.5mM 24 |
| | 3gr2 1.80 2009 2.52 Ki=3mM 24 |
| | 4kz6 1.68 2014 3.10 Ki=0.8mM 24 |
| | 4jxs 1.90 2014 4.74 Ki=18uM 24 |
| | 2r9w 1.80 2008 5.10 Ki=8uM 24 |
| | 2hb1 2.00 2006 3.80 Ki=160uM 25 |
| | 1bzc 2.35 1999 4.92 Ki=12uM 25 |
| | 2qbr 2.30 2008 6.33 Ki=0.47uM 25 |
| | 2qbq 2.10 2008 7.44 Ki=0.036uM 25 |
| | 2qbp 2.50 2008 8.40 Ki=0.004uM 25 |
| | 1q8t 2.00 2003 4.76 Kd=17.5uM 26 |
| | 1ydr 2.20 1997 5.52 Ki=3.0uM 26 |
| | 1q8u 1.90 2003 5.96 Kd=1.1uM 26 |
| | 1ydt 2.30 1997 7.32 Ki=48nM 26 |
| | 3ag9 2.00 2010 8.05 Ki=9nM 26 |
| | 3fcq 1.75 2009 2.77 Ki=1.7mM 27 |
| | 1z9g 1.70 2005 5.64 Ki=2.3uM 27 |
| | 1qf1 2.00 1999 7.32 Ki=48nM 27 |
| | 5tmn 1.60 1989 8.04 Ki=9.1nM 27 |
| | 4tmn 1.70 1989 10.17 Ki=0.068nM 27 |
| | 4ddk 1.75 2013 2.29 Kd=5.13mM 28 |
| | 4ddh 2.07 2013 3.32 Kd=0.48mM 28 |
| | 3ivg 1.95 2009 4.30 Kd=50uM 28 |
| | 3coz 2.00 2008 5.57 Kd=2.7uM 28 |
| | 3coy 2.03 2008 6.02 Kd=0.96uM 28 |
| | 3pxf 1.80 2011 4.43 Kd=37uM 29 |
| | 4eor 2.20 2013 6.30 Ki=500nM 29 |
| | 2xnb 1.85 2010 6.83 Ki=149nM 29 |
| | 1pxn 2.50 2004 7.15 Ki=0.07uM 29 |
| | 2fvd 1.85 2006 8.52 Ki=3nM 29 |
| | 4k77 2.40 2013 6.63 Ki=235nM 30 |
| | 4e5w 1.86 2012 7.66 Ki=22nM 30 |
| | 4ivb 1.90 2013 8.72 Ki=1.9nM 30 |
| | 4ivd 1.93 2013 9.52 Ki=0.3nM 30 |
| | 4ivc 2.35 2013 10.00 Ki=0.1nM 30 |
| | 4f09 2.40 2012 6.70 Ki=200nM 31 |
| | 4gfm 2.30 2013 7.22 Ki=0.06uM 31 |
| | 4hge 2.30 2012 7.92 Ki=11.9nM 31 |
| | 4e6q 1.95 2012 8.36 Ki=4.4nM 31 |
| | 4jia 1.85 2013 9.22 Ki=0.6nM 31 |
| | 2brb 2.10 2005 4.86 Ki=13.7uM 32 |
| | 2br1 2.00 2005 5.14 Ki=7.2uM 32 |
| | 3jvr 1.76 2009 5.72 Ki=1.89uM 32 |
| | 3jvs 1.90 2009 6.54 Kd=0.29uM 32 |
| | 1nvq 2.00 2003 8.25 Ki=5.6nM 32 |
| | 3acw 1.63 2010 4.76 Ki=17.5uM 33 |
| | 4ea2 2.05 2012 6.44 Ki=0.36uM 33 |
| | 2zcr 1.92 2008 6.87 Ki=135nM 33 |
| | 2zy1 1.78 2009 7.40 Ki=0.04uM 33 |
| | 2zcq 2.38 2008 8.82 Ki=1.5nM 33 |
| | 1bcu 2.00 1998 3.28 Kd=0.53mM 34 |
| | 3bv9 1.80 2008 5.36 Ki=4.4uM 34 |
| | 1oyt 1.67 2003 7.24 Ki=0.057uM 34 |
| | 2zda 1.73 2008 8.40 Ki=4nM 34 |
| | 3utu 1.55 2012 10.92 Ki=0.012nM 34 |
| | 3u9q 1.52 2011 4.38 Ki=41.7uM 35 |
| | 2yfe 2.00 2012 6.63 Ki=0.236uM 35 |
| | 3fur 2.30 2009 8.00 Ki=10nM 35 |
| | 3b1m 1.60 2011 8.48 Ki=3.3nM 35 |
| | 2p4y 2.25 2008 9.00 Ki=1nM 35 |
| | 3uo4 2.45 2012 6.52 Kd=299nM 36 |
| | 3up2 2.30 2012 7.40 Kd=40nM 36 |
| | 3e5a 2.30 2008 8.23 Ki=5.9nM 36 |
| | 2wtv 2.40 2010 8.74 Ki=1.8nM 36 |
| | 3myg 2.40 2010 10.70 Kd=0.02nM 36 |
| | 3kgp 2.35 2009 2.57 Ki=2.68mM 37 |
| | 1c5z 1.85 2000 4.01 Ki=97uM 37 |
| | 1o5b 1.85 2004 5.77 Ki=1.7uM 37 |
| | 1owh 1.61 2003 7.40 Ki=40nM 37 |
| | 1sqa 2.00 2004 9.21 Ki=0.62nM 37 |
| | 4jsz 1.90 2013 2.30 Ki=5000uM 38 |
| | 3kwa 2.00 2010 4.08 Ki=84uM 38 |
| | 2weg 1.10 2009 6.50 Kd=314nM 38 |
| | 3ryj 1.39 2011 7.80 Kd=16nM 38 |
| | 3dd0 1.48 2009 9.00 Ki=1nM 38 |
| | 2xdl 1.98 2010 3.10 Kd=790uM 39 |
| | 3b27 1.50 2011 5.16 Kd=6.9uM 39 |
| | 1yc1 1.70 2005 6.17 Kd=680nM 39 |
| | 3rlr 1.70 2011 7.52 Ki=30nM 39 |
| | 2yki 1.67 2011 9.46 Kd=0.35nM 39 |
| | 1z95 1.80 2005 7.12 Ki=76nM 40 |
| | 3b68 1.90 2008 8.40 Ki=4nM 40 |
| | 3b5r 1.80 2008 8.77 Ki=1.7nM 40 |
| | 3b65 1.80 2008 9.27 Ki=0.54nM 40 |
| | 3g0w 1.95 2009 9.52 Ki=0.3nM 40 |
| | 4u4s 1.90 2014 2.92 Kd=1200uM 41 |
| | 1p1q 2.00 2003 4.89 Kd=12.8uM 41 |
| | 1syi 2.10 2005 5.44 Ki=3590nM 41 |
| | 1p1n 1.60 2003 6.80 Kd=0.16uM 41 |
| | 2al5 1.65 2005 8.40 Ki=4nM 41 |
| | 3g2z 1.50 2009 2.36 Ki=4.4mM 42 |
| | 3g31 1.70 2009 2.89 Ki=1.3mM 42 |
| | 4de2 1.40 2012 4.12 Ki=76.0uM 42 |
| | 4de3 1.44 2012 5.52 Ki=3.0uM 42 |
| | 4de1 1.26 2012 5.96 Ki=1.1uM 42 |
| | 1vso 1.85 2007 4.72 Ki=18.98uM 43 |
| | 4dld 2.00 2012 5.82 Ki=1.5uM 43 |
| | 3gbb 2.10 2009 6.90 Ki=126nM 43 |
| | 3fv2 1.50 2010 8.11 Ki=7.7nM 43 |
| | 3fv1 1.50 2010 9.30 Ki=0.5nM 43 |
| | 4mgd 1.90 2014 4.69 Kd=20.19uM 44 |
| | 2qe4 2.40 2007 7.96 Ki=11.0nM 44 |
| | 1qkt 2.20 2000 9.04 Kd=0.92nM 44 |
| | 2pog 1.84 2007 9.54 Ki=0.29nM 44 |
| | 2p15 1.94 2007 10.30 Kd=50pM 44 |
| | 2y5h 1.33 2011 5.79 Ki=1620nM 45 |
| | 1lpg 2.00 2003 7.09 Ki=82nM 45 |
| | 2xbv 1.66 2010 8.43 Kd=3.7nM 45 |
| | 1z6e 1.80 2006 9.72 Ki=0.19nM 45 |
| | 1mq6 2.10 2003 11.15 Ki=7pM 45 |
| | 1nc3 2.20 2003 5.00 Ki=10uM 46 |
| | 1nc1 2.00 2003 6.12 Ki=0.75uM 46 |
| | 1y6r 2.20 2005 10.11 Ki=77pM 46 |
| | 4f2w 2.00 2013 11.30 Ki=5.0pM 46 |
| | 4f3c 1.93 2013 11.82 Ki=1.5pM 46 |
| | 1uto 1.15 2004 2.27 Kd=5.32mM 47 |
| | 4abg 1.52 2012 3.57 Kd=271uM 47 |
| | 3gy4 1.55 2010 5.10 Kd=8uM 47 |
| | 1k1i 2.20 2001 6.58 Kd=264nM 47 |
| | 1o3f 1.55 2003 7.96 Ki=0.011uM 47 |
| | 2yge 1.96 2011 5.06 Kd=8.62uM 48 |
| | 2fxs 2.00 2007 6.06 Kd=0.87uM 48 |
| | 2iwx 1.50 2006 6.68 Kd=0.21uM 48 |
| | 2wer 1.60 2009 7.05 Kd=90nM 48 |
| | 2vw5 1.90 2008 8.52 Kd=3nM 48 |
| | 4kzq 2.25 2013 6.10 Kd=788nM 49 |
| | 4kzu 2.10 2013 6.50 Ki=313nM 49 |
| | 4j21 1.93 2013 7.41 Kd=39nM 49 |
| | 4j3l 2.09 2013 7.80 Kd=16nM 49 |
| | 3kr8 2.10 2009 8.10 Kd=8nM 49 |
| | 2ymd 1.96 2012 3.16 Kd=693uM 50 |
| | 2wnc 2.20 2009 6.32 Kd=479nM 50 |
| | 2xys 1.91 2011 7.42 Ki=38nM 50 |
| | 2wn9 1.75 2009 8.52 Kd=3.0nM 50 |
| | 2x00 2.40 2010 11.33 Kd=4.7pM 50 |
| | 3ozt 1.48 2011 4.13 Ki=74.9uM 51 |
| | 3ozs 1.44 2011 5.33 Ki=4645nM 51 |
| | 3oe5 1.52 2011 6.88 Ki=132nM 51 |
| | 3oe4 1.49 2011 7.47 Ki=34nM 51 |
| | 3nw9 1.65 2011 9.00 Ki=1nM 51 |
| | 3ao4 1.95 2011 2.07 Kd=8.5mM 52 |
| | 3zt2 1.70 2012 2.84 Kd=1435uM 52 |
| | 3zsx 1.95 2012 3.28 Kd=519uM 52 |
| | 4cig 1.70 2014 3.67 Kd=214uM 52 |
| | 3zso 1.75 2012 5.12 Kd=7.6uM 52 |
| | 3n7a 2.00 2011 3.70 Ki=200uM 53 |
| | 4ciw 2.20 2014 4.82 Ki=15.0uM 53 |
| | 3n86 1.90 2011 5.64 Ki=2.3uM 53 |
| | 3n76 1.90 2011 6.85 Ki=0.14uM 53 |
| | 2xb8 2.40 2010 7.59 Ki=26nM 53 |
| | 4bkt 2.35 2013 3.62 Kd=240uM 54 |
| | 4w9c 2.20 2014 4.65 Kd=22.2uM 54 |
| | 4w9l 2.20 2014 5.02 Kd=9.52uM 54 |
| | 4w9i 2.40 2014 5.96 Kd=1.10uM 54 |
| | 4w9h 2.10 2014 6.73 Kd=0.185uM 54 |
| | 3nq9 1.90 2010 4.03 Kd=92.6uM 55 |
| | 3ueu 2.10 2011 5.24 Kd=5.81uM 55 |
| | 3uev 1.90 2011 5.89 Kd=1.29uM 55 |
| | 3uew 2.00 2011 6.31 Kd=0.49uM 55 |
| | 3uex 2.10 2011 6.92 Kd=0.12uM 55 |
| | 3lka 1.80 2010 2.82 Kd=1.5mM 56 |
| | 3ehy 1.90 2009 5.85 Ki=1.4uM 56 |
| | 3tsk 2.00 2012 7.17 Kd=67nM 56 |
| | 3nx7 1.80 2010 8.10 Kd=7.88nM 56 |
| | 4gr0 1.50 2013 9.55 Ki=0.28nM 56 |
| | 3dxg 1.39 2009 2.40 Ki=4.0mM 57 |
| | 3d6q 1.60 2009 3.76 Ki=172uM 57 |
| | 1w4o 1.60 2005 5.22 Ki=6uM 57 |
| | 1o0h 1.20 2003 5.92 Ki=1.2uM 57 |
| | 1u1b 2.00 2005 7.80 Kd=16nM 57 |
| |
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